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1-[(3-fluorophenyl)methyl]-4-[(quinolin-8-ylmethyl)amino]pyrrolidin-2-one
[(2,4-dimethoxy-3-methylphenyl)methyl](methyl)[(3-methyl-1H-pyrazol-4-yl)methyl]amine
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-2-(1-propylpiperidin-4-yl)acetamide
4-(4-fluorophenyl)-N-(isoquinolin-5-ylmethyl)-N-methyl-4-oxobutanamide
4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}benzamide
N-[2-(2H-1,3-benzodioxol-5-yl)pyridin-3-yl]cyclopropanecarboxamide
3-(1H-pyrazol-1-yl)-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]benzamide
[(5-ethylpyridin-2-yl)methyl](methyl)[(1-propyl-1H-imidazol-2-yl)methyl]amine
(2S,4S)-N-methyl-4-(4-{2-[(2,4,6-trimethylphenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
1-(2-chloroprop-2-en-1-yl)-3-{[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]methyl}-7-methyl-1,2-dihydroquinolin-2-one
6-methyl-2-[3-(1H-pyrazol-1-yl)phenyl]pyridine-3-carboxamide
1-(1,3-dihydro-2-benzofuran-5-yl)-3-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}urea
2-({[(3S,5S)-1-(2,3-dihydro-1H-inden-2-yl)-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-yl]amino}methyl)phenol
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanamide
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-5-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(1S,5R)-6-[5-(methoxymethyl)thiophene-2-carbonyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-2-(2-phenylethyl)-1,3-benzoxazole
2-(2-ethylphenyl)-N,N-dimethylpyridine-3-carboxamide
1-[3-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-(morpholin-4-yl)phenyl]ethan-1-one
4-[3-chloro-4-(1H-imidazol-1-yl)phenyl]-4H-1,2,4-triazole
(3aR,6aR)-2-(3-methylbenzenesulfonyl)-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-(4H-1,2,4-triazol-4-yl)benzamide
1-(cyclopropylmethyl)-4-{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}piperazine
2-(2,5-dimethylphenoxy)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
4-(benzyloxy)-1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
(3aS,6aS)-2-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N'-(4-methylphenyl)-N-[2-(quinolin-8-yloxy)ethyl]propanediamide
6-chloro-2-[2-(4-chlorophenyl)morpholin-4-yl]quinoline
8-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
9-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-(3-chlorophenyl)-N-(2-methoxyethyl)-N,7-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
8-[5-cyclopropyl-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]quinoline
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-3-(morpholin-4-yl)propanamide
1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
6-{[3-(piperidin-1-yl)pyrrolidin-1-yl]methyl}pyridine-2-carboxylic acid
N-benzyl-3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
7-{[4-(propan-2-yl)phenyl]methyl}-2-(thiophene-3-carbonyl)-2,7-diazaspiro[4.5]decane
3-(5-methylfuran-2-yl)-5-[2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]-1H-pyrazole
{3-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]phenyl}methanol
2-(5-chlorothiophen-2-yl)-4,6-dimethoxy-1,3,5-triazine
N-cyclopropyl-1-(3-methoxy-5-methylthiophene-2-carbonyl)piperazine-2-carboxamide
1-[6-(3-methylpiperidin-1-yl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
6-(1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)-2-methylpyrimidin-4-ol
N-benzyl-2-(2,6-dioxo-1,3-diazinan-1-yl)-N-[(4-fluorophenyl)methyl]acetamide
N-{2-[(2,4-dimethylphenyl)carbamoyl]ethyl}-4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]butanamide
1-[2-(2-hydroxyphenyl)acetyl]-3-methylpiperidine-3-carbonitrile
[(3,5-dichloropyridin-4-yl)methyl](methyl)(pyrazin-2-ylmethyl)amine
4-{4-[(2-ethylmorpholin-4-yl)methyl]phenyl}-2-methylbut-3-yn-2-ol
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]benzamide
N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-4-(pyridin-3-yloxy)piperidine-1-carboxamide