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[(2-chlorophenyl)methyl]({[2-(morpholin-4-yl)pyridin-3-yl]methyl})amine
2-[(2-methylprop-2-en-1-yl)oxy]-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
(4aS,7aR)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)(oxan-4-ylmethyl)amine
2-(cyclohex-3-en-1-yl)-1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1H-imidazole
[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl](methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
(4S,4aS,8aS)-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-phenyl-decahydroquinolin-4-ol
2-(3-fluorophenoxymethyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
dimethyl(2-{1-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-2-yl}ethyl)amine
(1S,5R)-3-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-3,9-diazabicyclo[3.3.2]decan-10-one
2-{[4-(morpholine-4-sulfonyl)piperazin-1-yl]methyl}-1H-1,3-benzodiazole
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-phenylpyrrolidin-3-ol
N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(1H-1,2,4-triazol-1-yl)acetamide
2-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]quinoline
(3aR,7aS)-2-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
(4aS,7aR)-1-[2-(piperidin-1-yl)acetyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)pyrimidine
3-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-methylurea
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-(methoxymethyl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[(3R,4R)-1-(1-benzothiophen-2-ylmethyl)-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
3-{[2-(furan-2-yl)ethyl]sulfamoyl}-N-(oxolan-2-ylmethyl)benzamide
N-(4-{4-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]piperidin-1-yl}phenyl)cyclopentanecarboxamide
4-[1-(methoxymethyl)cyclobutanecarbonyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-methyl-N-[1-(morpholin-4-ylmethyl)cyclopentyl]-1-propyl-1H-pyrazole-4-carboxamide
benzyl({[3-(pyrimidin-2-yloxy)phenyl]methyl})(1,3-thiazol-2-ylmethyl)amine
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-[7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-(4-methoxyphenoxy)ethan-1-one
3-[4-(4-fluorophenoxy)piperidine-1-carbonyl]-N,N-dimethylaniline
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-(methylsulfanyl)-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}propanamide
5-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-2-methylphenol
2-(1H-1,3-benzodiazol-1-yl)-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]acetamide
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-{[3-(methylsulfanyl)phenyl]methyl}butanamide
2-[4-(2-chloro-5-acetamidobenzoyl)morpholin-3-yl]acetic acid
methyl 5-[2-(2-oxopyrrolidin-1-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-(2-{[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]methyl}phenoxy)acetic acid
2-(2-phenyl-1,3-thiazol-4-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
1-[1-(2,5-difluorophenyl)cyclopropyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(2-methyl-1,3-benzothiazole-6-carbonyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
1-(1-cyclopropanecarbonylpiperidin-3-yl)-3-(3-fluoro-4-methylphenyl)urea
N-(1-carbamoylcyclopentyl)-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1,2-oxazole-3-carboxamide
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-(2-methoxyethyl)-N-methylacetamide
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)[(4,6-dimethylpyrimidin-2-yl)methyl]amine
N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(pyridin-4-yl)propyl]benzamide
{5-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
3-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
2-(1,1-dioxo-1λ6-thiomorpholin-4-yl)-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]benzamide
N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-3-(4H-1,2,4-triazol-4-yl)propanamide
dimethyl({[(2-phenoxypyridin-3-yl)methyl]sulfamoyl})amine
N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide