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3-(furan-2-yl)-2-[2-(2-phenyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]propanoic acid
(1-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]pyridin-2-yl}-3-ethylpiperidin-3-yl)methanol
N-(2-methylpropyl)-1-[(1s,4s)-4-(2,3,4-trimethoxybenzamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
methyl (2S,4S)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-[2-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
1-(propan-2-yl)-4-[4-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]pyrrolidin-2-one
4-(3-methylphenoxy)-1-(oxolane-3-carbonyl)piperidine
N-({3-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-[2-(6-methylpyridin-2-yl)ethyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[1-(1-benzyl-5-methyl-1H-1,2,3-triazole-4-carbonyl)piperidin-3-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-benzyl-8-(1,3-thiazol-4-ylmethyl)-2,8-diazaspiro[5.5]undecane
N-[2-(furan-2-yl)ethyl]-5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carboxamide
N-[(2-chlorophenyl)methyl]-N-cyclopropyl-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
3-[2-(dimethylamino)ethyl]-7-fluoro-3,4-dihydroquinazolin-4-one
N-(2,6-difluorophenyl)-2-(1,3-thiazol-2-yl)piperidine-1-carboxamide
2-{4-[5-(4-methoxyphenyl)furan-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-4-(1H-pyrazol-1-yl)butan-2-ol
(3aS,6aR)-5-benzoyl-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
9-[5-(4-methoxyphenyl)furan-2-carbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
1-[4-(1H-pyrazol-1-yl)phenyl]-N-[1-(pyridin-3-yl)propan-2-yl]piperidin-4-amine
3-[2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)ethyl]oxolan-2-one
5-(cyclohex-1-en-1-yl)-4,6-dimethyl-1H-pyrazolo[3,4-b]pyridin-3-amine
2-(4-acetylphenoxy)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
4-({4-[2-(azetidine-1-carbonyl)-4-methylphenoxy]piperidin-1-yl}methyl)pyridine
(1R,5R)-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(2S,4R)-N-(2-methoxyethyl)-1-(propan-2-yl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-(1-benzoylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
7-[(2,3-difluorophenyl)methyl]-2-(quinolin-8-ylmethyl)-2,7-diazaspiro[4.5]decane
[1-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)piperidin-4-yl]methanol
N4-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-N2,N2-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
2-(1-methyl-1H-indol-3-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
5-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidine-1-carbonyl]-2,1,3-benzoxadiazol-1-ium-1-olate
5-[3-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile
dimethyl({4-[1-(pyridazine-3-carbonyl)piperidin-2-yl]phenyl}methyl)amine
4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2,5,6-trimethylpyrimidine
3-[1-(2-methoxy-2-phenylacetyl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
1-(4-aminopyrimidin-2-yl)-3-(hydroxymethyl)piperidin-3-ol
N-benzyl-1-(3,5-dimethylfuran-2-carbonyl)-N-methylpiperidin-3-amine
3-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyridin-2-ol
N-{[7-methoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}-N-(3-methoxypropyl)thiophene-2-carboxamide
3-[2-(3-methoxypropyl)piperidine-1-carbonyl]-N,N-dimethylaniline
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-ethyl-4-{[1-(2-phenylethyl)piperidin-4-yl]amino}pyrrolidine-2-carboxamide
3-{methyl[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]sulfamoyl}-N-(propan-2-yl)benzamide
2-ethyl-N,N-bis(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
N-[4-(4-{[2-methyl-2-(morpholin-4-yl)propyl]amino}piperidin-1-yl)phenyl]benzenesulfonamide
4-{3-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]phenyl}-2-methylbutan-2-ol
3,5-dimethyl-2-({1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}methyl)-1,4-dihydropyridin-4-one
2-{[4-(2-fluorophenyl)-5-[(N-methylmethanesulfonamido)methyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-[1-(3-methylpentanoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
N-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,5-difluorobenzamide
2-(2-methoxyethyl)-8-[2-(pyrazin-2-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}quinoline-2-carboxamide