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methyl 4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]benzoate
N-[1-(4-{[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]oxane-4-carboxamide
methyl 2-(azocane-1-sulfonyl)-6-(1,2,3-thiadiazole-4-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-benzyl-4-(pyrimidin-2-yl)piperazine-1-sulfonamide
1-ethyl-4-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}piperazine
N-[(4-fluoro-2-methoxyphenyl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
9-(2-methoxypropanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
8-[(4-methoxy-2,5-dimethylphenyl)methyl]-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-({methyl[(3-phenyl-1,2-oxazol-5-yl)methyl]amino}methyl)-4H-chromen-4-one
(3S,7S)-5-(2,2-dimethylpropanoyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-(2H-1,3-benzodioxol-5-yl)-1-[2-(4-fluorophenyl)pyrrolidin-1-yl]ethan-1-one
N4-ethyl-N2-(1,2,2,6,6-pentamethylpiperidin-4-yl)pyrimidine-2,4-diamine
1-{5-[(2,6-difluorophenyl)methyl]-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-methyl-1,4-diazepane
1-(2-{4-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
(2-{4-[1-(dimethylamino)ethyl]phenyl}phenyl)methanol
3-[(3S,4R)-1-benzyl-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]-N-(oxolan-2-ylmethyl)propanamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({[3-oxo-3-(pyrrolidin-1-yl)propyl]amino}methyl)piperidin-2-one
N-methyl-N-(oxolan-3-yl)-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
2-amino-6-(2-hydroxypropan-2-yl)-4-(3-methyl-1-benzofuran-2-yl)pyridine-3-carbonitrile
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
1'-{[5-(2-fluorophenyl)furan-2-yl]methyl}-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(3S,4R)-1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N'-[(4-methoxyphenyl)methyl]-N-(5-methyl-1,2-oxazol-3-yl)-N'-(2-methylpropyl)ethanediamide
3-{2-oxo-2-[4-(pyrazin-2-yl)piperazin-1-yl]ethyl}-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidine-2,5-dione
[1-(1H-1,3-benzodiazol-2-yl)ethyl]({[3-chloro-5-methoxy-4-(prop-2-en-1-yloxy)phenyl]methyl})amine
4-(7-fluoro-2-methylquinoline-4-carbonyl)-N,N-dimethylpiperazine-1-carboxamide
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-4-(thiophen-2-yl)butanamide
N-cycloheptyl-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
(1S,5R)-3-[(2-propoxyphenyl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{[(1S,3R)-1-[2-(dimethylamino)ethoxy]-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]methyl}benzonitrile
4-(4-ethyl-1H-pyrazol-5-yl)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidine
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)imidazo[1,2-b]pyridazine-3-carboxamide
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N,5-dimethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]thieno[2,3-d]pyrimidine-6-carboxamide
3-(2-fluorophenyl)-N-[(3-methylpyridin-2-yl)methyl]-3-phenylpropanamide
N-[2-(7-methyl-1H-indol-3-yl)ethyl]-2-(pyrrolidin-3-yl)acetamide
7-[2-(phenylamino)pyrimidine-5-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
{3-[(3-methoxyphenyl)methyl]-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl}methanol
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-5-chloro-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-2,6-dimethylphenol
N,1-dimethyl-6-oxo-N-[1-(3-phenylpropyl)piperidin-3-yl]-1,4,5,6-tetrahydropyridazine-3-carboxamide
4-(4-methanesulfonylphenyl)-6-(pyrrolidin-1-yl)pyrimidin-2-amine
N-[(5-fluoro-1H-indol-2-yl)methyl]-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
4-(azocan-1-yl)-N-butyl-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
2-{2-[(3R)-3-hydroxypyrrolidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
5-{[benzyl(methyl)amino]methyl}-N-[(2,6-difluorophenyl)methyl]-1,2-oxazole-3-carboxamide
2-{1-[3-methyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]propyl}-2,3-dihydro-1H-isoindol-1-one
5-[3-(propoxymethyl)pyrrolidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidin-4-ol
1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-4-(thian-4-yl)piperazine
2-(1H-imidazol-1-yl)-1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide