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N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
7-(propan-2-yl)-2-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-2,7-diazaspiro[4.5]decan-6-one
1-[(4-methyloxan-4-yl)methyl]-4-phenylpiperidine-4-carbonitrile
1-{2-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-3-methyl-1,2-dihydroquinoxalin-2-one
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]acetamide
N-[(3-methylphenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
1-{5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
1-[4-(3-chlorophenyl)-2-methyl-5-oxopiperazine-1-carbonyl]cyclopropane-1-carboxamide
(4aS,7aR)-1-[(3E)-pent-3-enoyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S)-2-phenyl-2-[2-(2,5,7-trimethyl-1H-indol-3-yl)acetamido]acetamide
1-(2-{1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
2-(2-hydroxyethyl)-9-(4-methoxypyrimidin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-(4-ethenylbenzoyl)-2-[(3-methoxyphenyl)methyl]morpholine
2-{1-[(2-fluorophenyl)methyl]-4-(9H-purin-6-yl)piperazin-2-yl}ethan-1-ol
N-(4-acetylphenyl)-3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carboxamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-{4-[6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-1H-pyrazol-1-yl}acetamide
6-[9-acetyl-7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]pyridine-3-carboxamide
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
3-(2,6-difluorophenyl)-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
N-[1-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]oxolane-3-carboxamide
3-[2-(2,6-difluorophenyl)ethyl]-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N,5-dimethyl-1H-pyrazole-3-carboxamide
N-(8-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-{1-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
5,6-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-oxo-1,2-dihydropyridine-3-carboxamide
4-amino-2-[4-(pyrimidin-5-ylmethyl)piperazin-1-yl]pyrimidine-5-carbonitrile
(3S,9aR)-8-[(2,4-dimethylphenyl)methyl]-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{2-[4-(cyclopropylmethyl)morpholin-2-yl]ethyl}-5-methylpyridine-3-carboxamide
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)piperidine-3-carboxamide
8-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
5-[1-(oxan-4-yl)piperidine-4-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-oxo-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-2,3-dihydro-1H-indene-1-carboxamide
1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
3-ethyl-8-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(4-methylphenoxymethyl)-1-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-ethyl-5-[2-(3-phenylpropyl)morpholine-4-carbonyl]pyrimidin-2-amine
{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amine
1-[(2,4-dimethoxyphenyl)methyl]-4-(2-methylquinolin-6-yl)piperidin-4-ol
N-(2-{[3-(3-methoxyphenyl)-1H-pyrazol-4-yl]formamido}ethyl)pyridine-3-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-(1,3-thiazole-4-carbonyl)piperidine-4-carboxylate
2-methoxy-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}pyridine-3-carboxamide
3-[(3R,4S)-1-(4,6-dimethylpyridine-3-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(3R,5S)-N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
1-methyl-2-[3-(pyridin-2-yl)azetidine-1-carbonyl]azepane
9-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-{4-[3-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-6-(2-methoxyphenyl)pyridine-3-carboxamide
2-(4-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-1-(furan-2-ylmethyl)piperazin-2-yl)ethan-1-ol