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1-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
1-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-[2-methyl-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
6-methyl-N-[1-(methylcarbamoyl)cyclohexyl]imidazo[1,2-a]pyridine-2-carboxamide
1-[(4-fluoro-3-methoxyphenyl)methyl]-3-(pyrrolidin-1-yl)piperidine
2-{1-[(1-cyclopentylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}pyridine
6-[4-(2-fluoro-4-methanesulfonylphenyl)piperazin-1-yl]-N,N-dimethylpyrimidin-4-amine
(3R,4R)-1-[(9-ethyl-9H-carbazol-3-yl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
2-({[(3R,4R)-1-[(2,6-dichlorophenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[2-(pyridin-2-yl)ethyl]-3-{[(3R)-pyrrolidin-3-yl]sulfamoyl}benzamide
6-{1-[(2-aminopyridin-3-yl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-({[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)piperidin-2-one
4-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]pyrrolidin-2-one
4-(2-benzyl-3-oxopiperazine-1-carbonyl)benzonitrile
2-(1-methyl-1H-1,3-benzodiazol-2-yl)-N-(prop-2-en-1-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
3,7-dimethyl-11-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}-3,7,11-triazaspiro[5.6]dodecane
N-benzyl-6-oxo-N-(1,3-thiazol-2-ylmethyl)-1,6-dihydropyridine-3-carboxamide
(1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-phenylethyl)(2-methoxyethyl)(pyridin-2-ylmethyl)amine
1-[(4-fluorophenyl)methyl]-3-{2-[(3S)-3-hydroxypyrrolidin-1-yl]-2-oxoethyl}-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
(4aS,8aS)-4a-hydroxy-N-(3-phenyl-1,2,4-thiadiazol-5-yl)-decahydroisoquinoline-2-carboxamide
6-[1-(4-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
2,8-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]quinoline-4-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-1-[1-(furan-2-ylmethyl)piperidin-4-yl]piperidin-3-amine
4-{[4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
4-(1H-pyrazol-1-yl)-2-[4-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]butan-2-ol
methyl 6-cyclopentanecarbonyl-2-[(2,3-dimethylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(2-chloro-3-methoxyphenyl)-3-methyl-3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}urea
5-(1H-indol-1-ylmethyl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methyl-N-(2-phenylethyl)piperidine-1-carboxamide
5-[(1,3-benzothiazol-2-ylmethyl)(methyl)amino]-N-benzyl-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
6-(propan-2-yl)-N-[1-(thiophene-2-carbonyl)piperidin-3-yl]pyrimidin-4-amine
N-(4-fluoro-3-methoxyphenyl)-4-(pyrrolidine-1-carbonyl)piperidine-1-carboxamide
6-[2-(aminomethyl)-5-fluoro-2,3-dihydro-1-benzofuran-7-yl]isoquinolin-3-amine
1-(2-methoxyethyl)-3-[3-(2,2,2-trifluoroethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrrolidine
(3S,4R)-4-(3-methoxyphenyl)-1-[2-(methylsulfanyl)pyridine-3-carbonyl]pyrrolidine-3-carboxylic acid
3-[(methylsulfanyl)methyl]-5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1,2,4-oxadiazole
2-chloro-5-({[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]carbamoyl}amino)-N-methylbenzamide
2-amino-4-[3-(ethoxymethyl)-4-methoxyphenyl]-6-ethyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-{2-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]-2-oxoethyl}piperidin-2-one
2-ethyl-N-[1-(thiophen-2-yl)butyl]pyrimidine-5-carboxamide
(3R,4R)-1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3,4-dimethylpyrrolidin-3-ol
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-cyclobutylpiperidine-3-carboxamide
(3S,4S)-4-(pyridin-2-yl)-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]pyrrolidine-3-carboxylic acid
N-ethyl-N-methyl-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrimidin-4-amine
[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl){[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
(1S,5R)-3-(4-cyclopentylpyrimidin-2-yl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-benzyl-5-[4-(hydroxymethyl)piperidin-1-yl]-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(2,3-difluoro-4-methoxyphenyl)methyl]-4-(piperidin-1-ylmethyl)piperidine
N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-1-(trifluoromethyl)cyclopropane-1-carboxamide
4-(2-methylpropyl)-1-[3-(pyridin-3-yl)propyl]pyrrolidin-2-one