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(2S,4R)-4-amino-N-methyl-1-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}pyrrolidine-2-carboxamide
N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]quinoline-8-carboxamide
2-(3-methoxypropyl)-8-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
2-amino-4-(3-chlorophenyl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-2-carboxamide
4-(4-{[(3-fluorophenyl)methyl]amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
(2S,4S)-4-amino-N,N-diethyl-1-(1,8-naphthyridine-2-carbonyl)pyrrolidine-2-carboxamide
1-{2-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazine-1-carboxylate
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(thiophen-2-ylmethyl)piperidin-3-yl]propanoic acid
[3-({1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]pyrrolidin-3-yl}methyl)phenyl]methanol
8-(2-aminopyridine-4-carbonyl)-2-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(3-methylphenyl)-1-[3-(1H-pyrazol-1-yl)benzoyl]piperidine
3-methyl-4-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
5-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1,3-oxazole-4-carboxamide
1-ethyl-4-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)-1H-indole
N-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}pyrazin-2-amine
2-(morpholin-4-ylmethyl)-4-[(1-propyl-1H-imidazol-2-yl)methyl]-1,4-oxazepane
3-{[(2S,4S)-4-fluoro-1-[2-(methylsulfanyl)acetyl]pyrrolidin-2-yl]methyl}-1-methyl-1-phenylurea
4-fluoro-2-{[(isoquinolin-5-ylmethyl)(methyl)amino]methyl}phenol
4-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)-1,4-diazepane-1-carbaldehyde
2-methyl-N-[2-(3-methylthiophen-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-N-methylpyridine-3-carboxamide
dimethyl(1-{1-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]piperidin-4-yl}ethyl)amine
1,4-dimethyl 2-({1-[4-(pyrazine-2-amido)phenyl]piperidin-4-yl}amino)butanedioate
[(3S,4S)-4-(hydroxymethyl)-1-[6-(propan-2-yl)pyrimidin-4-yl]pyrrolidin-3-yl]methanol
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-2,1-benzoxazole-3-carboxamide
3-[4-(5-{[(2-methoxyphenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidin-1-yl]propanamide
1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-(pyridin-3-yl)piperazine
6-ethyl-2-(3-{[methyl(oxolan-2-ylmethyl)amino]methyl}phenyl)-3H,4H,5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-one
(1s,4s)-4-[4-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexan-1-amine
5,6-dimethyl-N-[(4-methyl-1,4-oxazepan-6-yl)methyl]-2-(trifluoromethyl)pyrimidin-4-amine
4-(4-fluorophenyl)-2-(morpholin-4-ylmethyl)phenol
1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-3-phenylpiperazine
2-[(4-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carbonyl}phenyl)sulfanyl]ethan-1-ol
1-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
(2S,4R)-N-[2-(2-fluorophenyl)ethyl]-4-({[4-(methylsulfanyl)phenyl]methyl}amino)-1-(propan-2-yl)pyrrolidine-2-carboxamide
6-ethyl-N,2-dimethyl-N-[2-(1H-pyrazol-4-yl)ethyl]quinoline-4-carboxamide
1-(2-methoxypyridine-3-carbonyl)-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
1-(2-ethylphenyl)-4-[1-(2-methoxyethyl)piperidine-3-carbonyl]piperazine
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(2-methoxyacetyl)pyrrolidin-3-yl]-5-methyl-1,3-oxazole-4-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(prop-2-en-1-ylsulfanyl)propan-1-one
4-(1-hydroxy-3-phenylpropyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
1-[4-(1H-imidazol-1-ylmethyl)phenyl]-3-methyl-1H-pyrazole
1-(2-{[(5-phenyl-1,3,4-thiadiazol-2-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
(2S,4R)-4-amino-N-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}pyrrolidine-2-carboxamide
(4aR,8aR)-4a-hydroxy-7-[(2-methoxypyridin-3-yl)methyl]-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
2-acetyl-8-(thiophene-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
8-[5-fluoro-2-(hydroxymethyl)pyridin-4-yl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid