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1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(methoxymethyl)-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
ethyl 1-(2-methyl-1-benzofuran-5-carbonyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
5-{3-[4-(4-methoxyphenyl)-3-oxopiperazin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
2-[4-(1-methoxypropan-2-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
6-methoxy-1-methyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1H-indole-2-carboxamide
4-(azepane-1-carbonyl)-8-methyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
N-[2-(4-fluorophenyl)ethyl]morpholine-2-carboxamide
(4S)-1-{5-[(dimethylamino)methyl]furan-2-carbonyl}-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
2-cyclopropyl-4-[3-(4-phenylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
3-(morpholin-4-yl)-N-(1-phenylbutyl)benzamide
1-{4-[(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)methyl]thiophen-2-yl}ethan-1-one
1-(1-benzylpyrrolidin-3-yl)-5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)pyrrolidin-2-one
N-(6-methoxyquinolin-8-yl)-6-oxa-9-azaspiro[4.5]decane-9-carboxamide
{[4-(butan-2-yloxy)-3-methoxyphenyl]methyl}({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amine
2-methyl-4-{[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-imidazole
4-[2-(3-benzoylpiperidin-1-yl)pyridine-4-carbonyl]morpholine
1-(3,5-dimethylphenyl)-4-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperazin-2-one
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(4-methyl-1H-pyrazol-1-yl)propanamide
7-(propan-2-yl)-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(oxolan-2-ylmethyl)amine
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,2-oxazole-3-carbonyl)piperidine
N-(4-chloro-3-methylphenyl)-2-[cyclopropyl(1,3-thiazol-5-ylmethyl)amino]acetamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(2-methylpropyl)amino]methyl}piperidin-2-one
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
2-(4-fluorophenyl)-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)acetamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
5,7-dimethyl-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
N3-[2-(3,4-dimethoxyphenyl)ethyl]-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-methyl-4-{1-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]ethyl}piperazine
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]amine
(2S,4R)-4-(cyclooctylamino)-N-methyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[2-(pyrazin-2-yl)ethyl]pyridin-2-amine
3-ethyl-1-{2-[4-(methylsulfanyl)phenyl]acetyl}piperidine-3-carboxylic acid
2-{methyl[1-(1,2-oxazol-3-yl)ethyl]amino}-N-(pyrazin-2-yl)acetamide
2-methyl-1-{2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}-1H-imidazole
1-[4-methyl-7-(methylsulfanyl)quinolin-2-yl]butan-2-ol
N-{4-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)acetamido]-2-methoxyphenyl}butanamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-N,2,6-trimethylpyridine-4-carboxamide
2-[(2-methylprop-2-en-1-yl)oxy]-N-(2-propoxyethyl)benzamide
(2S,4R)-4-({[4-(methylsulfanyl)phenyl]methyl}amino)-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1-(propan-2-yl)piperidine-4-carboxamide
4-{2-methoxy-5-[3-(methoxymethyl)pyrrolidine-1-carbonyl]phenoxy}-1-(propan-2-yl)piperidine
N-(1,3-benzothiazol-2-ylmethyl)-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(4-{[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenyl)prop-2-yn-1-ol
3-(1-methyl-1H-imidazol-2-yl)-6-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}pyridazine
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-2-(thiophen-2-yl)-1,3-thiazole
8-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-2-cyclopentyl-2,8-diazaspiro[5.5]undecan-3-one
(1H-1,3-benzodiazol-5-ylmethyl)(methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
1-methyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]azepane-2-carboxamide