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1-({5-[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]furan-2-yl}methyl)-4-methylpiperazine
4-({[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl)amino}methyl)benzonitrile
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-({[2-(pyridin-2-yl)ethyl]amino}methyl)piperidin-2-one
3-(3-hydroxypropyl)-5-[(3-methoxyphenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
N-[3-(pyridin-3-yl)propyl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
N-cyclobutyl-3-(3-hydroxy-3-methylbutyl)benzamide
4-benzyl-3-[1-(cyclopropylmethyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazole
1-ethyl-N-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(3-chlorophenyl)methyl]-3-[1-(furan-2-carbonyl)piperidin-4-yl]propanamide
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N,1-dimethyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
6-{[4-(morpholin-4-yl)piperidin-1-yl]methyl}-1H-indole
2-(2-ethoxyacetyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)benzamide
2-methoxy-4-[({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)methyl]phenol
ethyl 1-[(2-ethoxy-2-oxoethyl)carbamoyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
2-(dimethylamino)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(3-methylphenyl)ethan-1-one
N-(3-chloro-4-methoxyphenyl)-6-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
(4aS,7aR)-1-(1-methyl-1H-pyrrole-2-carbonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]propane-1,2-diol
8-methyl-2-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-2,8-diazaspiro[4.5]decane
4-[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]pyrimidine-5-carboxylic acid
N-cyclopentyl-1-{1-[(4-acetamidophenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
(benzylsulfamoyl)({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl})amine
2-methoxy-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
N-cyclopropyl-3-[5-(pyridine-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-{2-[4-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,3-oxazinan-2-one
1-cyclopentanecarbonyl-N-[2-(4-fluorophenyl)-2-hydroxyethyl]piperidine-4-carboxamide
N-{[5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
1-(2,3-dihydro-1-benzofuran-2-carbonyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine
2-{1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1,4-diazepan-6-yl}acetic acid
N'1-methyl-N'1-[3-(pyrrolidin-1-yl)butyl]cyclopropane-1,1-dicarboxamide
2-(3-chloropyridin-2-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
(2S,4R)-1-benzyl-4-{[(3-chlorophenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-({3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]phenyl}formamido)acetamide
7-(3-chlorophenyl)-4-(furan-2-ylmethyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{[3-(methylsulfanyl)phenyl]methyl}-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
2-{[(2-methylpropyl)amino]methyl}-4-(pyridin-3-yl)phenol
ethyl 2-({5-[2-amino-3-cyano-6-(5-methylfuran-2-yl)pyridin-4-yl]pyrimidin-2-yl}amino)acetate
5-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
methyl 4-(3-{[3-(3-methylphenyl)phenyl]carbamoyl}piperidin-1-yl)-4-oxobutanoate
2-[(3-chlorophenyl)methyl]-N-[3-(pyridin-3-yl)propyl]-1,3-benzoxazole-6-carboxamide
2-[5-(6-cyanopyridin-3-yl)-1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-3-yl]acetamide
2-(3-methyl-1,2-oxazol-5-yl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N-(1H-indazol-5-yl)-1-methylpyrrolidine-3-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)-N-(propan-2-yl)acetamide
N-[(1R,3R)-3-aminocyclopentyl]-1-tert-butyl-1H-pyrrole-3-carboxamide
2-(3-methoxyphenoxy)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one