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2-(5-phenyl-1,3,4-thiadiazol-2-yl)-1,2,3,4-tetrahydroisoquinolin-4-ol
2-(1,2-benzoxazol-3-yl)-N-{[6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidin-4-yl]methyl}acetamide
4-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-1,4-oxazepan-5-one
2-(3-methoxyphenyl)-N-[(5-methylthiophen-2-yl)methyl]acetamide
4-(furan-3-ylmethyl)-3-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-oxoethyl]piperazin-2-one
1-(2-ethoxyethyl)-5-(4-ethylpiperazine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-[4-(3-hydroxy-3-methylbutyl)benzoyl]piperidine-3-carbonitrile
5-(3-benzoylpiperidine-1-carbonyl)-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
N-[2-(dimethylsulfamoyl)ethyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N2,N2,N4,N4-tetramethyl-7-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
3-(2H-1,3-benzodioxol-5-yl)-2-methoxypyridine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-methyl-2-(methylamino)-1,3-thiazole-5-carboxamide
2-[1-({1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
(1S,5R)-N-(2-methoxyphenyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
1-(1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-4-phenylpiperidin-4-yl)ethan-1-one
N-{4-[3-(2-methoxyphenoxy)azetidin-1-yl]-4-oxobutyl}acetamide
5-{2-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
3-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]benzonitrile
1-{4-[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]piperidin-1-yl}ethan-1-one
6-(azocane-1-carbonyl)-5-methyl-N-(oxolan-2-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
[(2S,6S)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
5-(1H-indol-1-ylmethyl)-N-[1-(pyrazin-2-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
4-(1,4-dithiepan-6-yl)-N-[2-(pyridin-2-yl)ethyl]morpholine-2-carboxamide
2-ethyl-9-(pyrimidin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-{2-oxo-8-[2-(1H-pyrrol-1-yl)pentanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetic acid
2-({[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)amino)ethan-1-ol
N-benzyl-2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
methyl 2-(4-{[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}piperidin-1-yl)acetate
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-4-ylmethyl)acetamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
N-(3-butanamidophenyl)-3-hydroxy-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
4-[3-(morpholine-4-carbonyl)piperidin-1-yl]-N-propylpiperidine-1-carboxamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(pyridin-4-yl)propanamide
N-({1-[(2-cyanophenyl)methyl]pyrrolidin-3-yl}methyl)but-3-enamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(1-methyl-1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
3-{[(4-fluorophenyl)methyl]amino}-N-methyl-N-[(1-methylpyrrolidin-3-yl)methyl]benzamide
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
3-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-[2-methoxy-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
2-{4-[2,5-dioxo-4-(pyridin-2-yl)imidazolidin-4-yl]piperidin-1-yl}-6-methylpyridine-3-carbonitrile
ethyl 4-[(3-fluorophenyl)methyl]-1-[2-(methylsulfanyl)acetyl]piperidine-4-carboxylate
1-benzyl-5-(furan-2-yl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-1H-1,3-benzodiazole-2-carboxamide
3-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[2-(methylsulfanyl)ethyl]benzamide
N-(furan-3-ylmethyl)-7-methoxy-N,4-dimethylquinazolin-2-amine
2-[(4-benzylpiperazin-1-yl)methyl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(pyridin-2-yl)ethan-1-one
2-[(5-{2-amino-3-cyano-5H,6H-benzo[h]quinolin-4-yl}pyrimidin-2-yl)amino]acetic acid
N-[3-(propan-2-yloxy)propyl]-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide