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4-(1-butyl-1H-imidazol-2-yl)-1-[(4-methanesulfonylphenyl)methyl]piperidine
N-(2-methylpropyl)-1-[1-(pent-4-enoyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
N-[3-({[2-(azepan-1-yl)ethyl]carbamoyl}amino)-4-chlorophenyl]-2-methoxyacetamide
N-(6-fluoropyridin-3-yl)-4-(2-phenylethyl)piperazine-1-carboxamide
1-methyl-4-{2-[4-(pyridin-4-yl)piperidin-1-yl]pyridine-4-carbonyl}piperazine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(3-methyl-1,2-oxazol-5-yl)acetamide
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-5-(methoxymethyl)furan-2-carboxamide
3-(2,3-dimethoxyphenyl)-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)pyrrolidine
1-[2-methyl-4-(morpholin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
6-(1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)-2-methylpyrimidin-4-ol
4-cyclopropanecarbonyl-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
ethyl 1-{[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-4-carboxylate
N-{4-[2-amino-3-cyano-6-(4-hydroxyphenyl)pyridin-4-yl]phenyl}acetamide
2-amino-4-(1H-imidazol-4-yl)-5H,6H-furo[2,3-h]quinoline-3-carbonitrile
4-[(5-methylfuran-2-yl)methyl]-3-{[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-2-one
2-(1H-imidazol-2-yl)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}benzamide
2-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-4-carboxamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]-1-cycloheptyl-1H-1,2,3-triazole-4-carboxamide
(1S,2R)-2-({[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}(methyl)amino)cyclohexan-1-ol
N-methyl-2-[4-(propan-2-yl)morpholin-2-yl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
4-(2,4-dioxoimidazolidin-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
2-[(3,4-dimethoxypyridin-2-yl)methyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
N-[3-(2-chlorophenoxy)propyl]-2-(2,6-dioxo-1,3-diazinan-1-yl)-N-methylacetamide
4-[(2-hydroxyethyl)(methyl)amino]-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzamide
N-methyl-2-(1H-pyrazol-1-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]acetamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-5-(2-methylphenyl)-1,2,4-triazin-3-amine
diethyl({3-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3-fluorophenyl)ethan-1-one
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-5-(propan-2-yl)pyrimidine
8-fluoro-N-[(5-methyl-1,2-oxazol-3-yl)methyl]quinoline-2-carboxamide
N3-[2-(3-fluorophenyl)ethyl]-4-oxo-1-(oxolan-2-ylmethyl)-N5-(2,2,2-trifluoroethyl)-1,4-dihydropyridine-3,5-dicarboxamide
3-[5-(4-fluorophenoxymethyl)-3-(furan-2-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
(1s,4s)-4-{[4-(2-methylphenyl)-1,4-diazepan-1-yl]methyl}cyclohexan-1-amine
5-methoxy-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]furan-2-carboxamide
3-bromo-5-[(oxolan-2-ylmethyl)sulfamoyl]benzoic acid
4-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-1-(3-methoxyphenyl)piperazin-2-one
N,3,5-trimethyl-N-(quinoxalin-6-ylmethyl)-1H-indole-2-carboxamide
[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl})methylamine
N-cyclopentyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
4-ethyl-3-({1-[(2S)-2-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2R)-2-amino-1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
2-{2-[6-amino-5-cyano-4-(furan-2-yl)pyridin-2-yl]phenoxy}acetamide
4-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethyl]-1-phenyl-3-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-phenyl-N-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1,3-thiazole-2-carboxamide
6-amino-N-methyl-N-[(4-phenoxyphenyl)methyl]pyridine-3-carboxamide
14-(pentan-3-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
(2S)-1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-[2-(morpholin-3-yl)acetamido]thieno[2,3-b]pyridine-2-carboxylic acid
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1H-indazol-1-yl)acetamide