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N-{1-[4-(3-chlorophenyl)-5-[(cyclohexylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}pent-4-enamide
2-[3-(aminomethyl)piperidine-1-carbonyl]-N-methyl-N-(2-phenylethyl)-2,3-dihydro-1H-inden-2-amine
1-[(4aR,8aR)-1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-2-(2-methoxyphenyl)ethan-1-one
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]pyrimidine-5-carboxamide
N-{1-[1-(2,3-difluorobenzoyl)piperidin-4-yl]-2-phenylethyl}-N-methylpyridine-2-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[4-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methanol
1-[1-({2-oxo-3-oxatricyclo[7.3.1.05,13]trideca-1(12),5(13),6,8,10-pentaen-8-yl}methyl)piperidin-3-yl]pyrrolidin-2-one
2-methoxy-4-[(1E)-3-[3-(morpholin-4-yl)piperidin-1-yl]prop-1-en-1-yl]phenol
1-[4-(2-methoxybenzoyl)piperazin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
(1R,5R)-6-(cyclobutylmethyl)-3-{pyrazolo[1,5-a]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
2-amino-5-methyl-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
N-[4-fluoro-3-(trifluoromethyl)phenyl]-2,8-diazaspiro[4.5]decane-2-carboxamide
N-[(3R,4R)-3-hydroxy-1-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]piperidin-4-yl]pyridine-3-carboxamide
2-[1-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-ol
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-1-(4-methylpiperidin-1-yl)ethan-1-one
5-chloro-2-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1,2,3,4-tetrahydroisoquinoline
4-{1-[(5-chlorofuran-2-yl)methyl]piperidin-3-yl}pyrimidine
3-(2,3-dihydro-1-benzofuran-7-yl)-5-(morpholine-4-sulfonyl)benzoic acid
2-(dimethylamino)-8-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
4-(2-methoxyacetyl)-N-[2-methyl-3-(pyrrolidin-1-yl)phenyl]-1,4-diazepane-1-carboxamide
N-({3-[(1-cyclohexanecarbonylpiperidin-3-yl)methoxy]phenyl}methyl)-N,1-dimethylpiperidin-4-amine
1-methyl-3-(propan-2-yl)-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-1H-pyrazole-5-carboxamide
N-[1-(6-methoxynaphthalen-2-yl)ethyl]-2-[methyl(piperidin-4-yl)amino]acetamide
2-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-4-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-4-(pyridin-3-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
2-[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidin-4-yl]acetamide
N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N-[5-({[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]carbamoyl}amino)-2-fluorophenyl]-2-methylpropanamide
1-[(1-{6-[4-(hydroxymethyl)phenyl]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
4-[(2,6-dimethylpyridin-3-yl)oxy]-1-(pyridin-4-yl)piperidine-4-carboxylic acid
N-(2,3-dihydro-1-benzofuran-3-yl)-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
{3-[(4-fluorophenyl)methyl]-1-(6-methylpyridazin-3-yl)piperidin-3-yl}methanol
2-{4-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}-4-(thiophen-2-yl)pyrimidine
(2-methoxyethyl)[(4-methylphenyl)methyl](quinoxalin-2-ylmethyl)amine
2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-1-(pyrrolidin-1-yl)propan-1-one
4-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
2-amino-1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
(3S,4S)-1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-4-propylpyrrolidine-3-carboxylic acid
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-[2-(1H-imidazol-2-yl)benzoyl]-3-(pyrrolidine-1-carbonyl)piperidine
8-(2-ethylpyrimidine-5-carbonyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
7-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-2-oxa-7-azaspiro[4.5]decan-8-one
1-(4-benzylpiperidin-1-yl)-3-[1-(5-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]propan-1-one
4-{4-[(1,4-dioxan-2-ylmethyl)(methyl)amino]piperidin-1-yl}-N-[2-(morpholin-4-yl)ethyl]benzamide
3-butyl-4-(3-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one