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3-{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidine-3-carbonyl}pyridine
2-({[(3R,4R)-4-(hydroxymethyl)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-(4-fluorophenyl)-4-[1-(pyridine-4-carbonyl)piperidin-3-yl]piperazine
N-ethyl-2-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]pyrimidin-4-amine
methyl 5-(cyclobutylamino)-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-methyl-N-[2-(1-methyl-1H-pyrrol-2-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
3-{[2-({2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]methyl}pyridin-2-amine
9-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-methyl-8-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 3-(4-methoxybenzamido)-1-methyl-5-[(4,4,4-trifluorobutan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3-methyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
4-{1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-3-phenyl-1H-pyrazole
3-methyl-7-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
{3-[(2-fluorophenyl)methyl]-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl}methanol
5-(furan-2-yl)-3-{[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2-oxazole
1-cyclopentyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]piperidine-3-carboxamide
N-[2-(3-fluorophenyl)ethyl]-2-(4-{4-[(1-methoxypropan-2-yl)amino]piperidin-1-yl}phenyl)acetamide
2-chloro-4-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}benzamide
(1R,5R)-3-benzoyl-6-[(3-chloro-2-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-[(2-amino-6-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidin-4-yl)amino]ethan-1-ol
1-(2,3-dihydro-1H-inden-2-yl)-N-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
methyl 6-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1,9-dimethyl-4-(2-methylpyrimidin-4-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[4-(2,1,3-benzothiadiazol-4-yl)-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl]methanesulfonamide
4-benzyl-1-[(dimethyl-1,2-oxazol-4-yl)methyl]pyrrolidin-2-one
2-ethyl-8-{2-[(3-methoxyphenyl)sulfanyl]acetyl}-2,8-diazaspiro[5.5]undecan-3-one
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-benzyl-N-[2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]pyrrolidin-3-amine
1-{6-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]pyridin-2-yl}ethan-1-ol
N-(1H-imidazol-2-ylmethyl)-N-methyl-3-(2-methylphenyl)benzamide
1-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
8-(2-methoxyethyl)-N-methyl-9-oxo-N-phenyl-2,8-diazaspiro[5.5]undecane-2-carboxamide
N-methyl-N-(1,2-oxazol-3-ylmethyl)-2-phenylbenzamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[2-(pyrazin-2-yl)ethyl]benzamide
1-(3-methylbutyl)-3,8-bis(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1-cycloheptylpiperidin-3-yl)-2-(3-methyl-1H-pyrazol-1-yl)acetamide
2-(cyclopropylmethyl)-N-(4-fluorophenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2,6-dimethylquinoline-3-carboxamide
5-(2-methoxyphenoxymethyl)-N-methyl-N-[1-(pyridin-4-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[(3S,4R)-1-(2,6-dimethoxypyridine-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
5-(4-acetylphenoxymethyl)-N-ethyl-N-[2-(pyrrolidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
(2S)-1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
8-chloro-2-{[2-(trifluoromethyl)morpholin-4-yl]methyl}quinoline
1-(cyclohexylmethyl)-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]furan-2-carboxamide
1-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
1-[(4-chlorophenyl)methyl]-N-(3-hydroxy-3-methylbutyl)-N-methyl-6-oxopiperidine-3-carboxamide
N-(3-hydroxy-3-phenylpropyl)-N-methyl-5-(morpholin-4-ylmethyl)furan-3-carboxamide
2-(dimethylamino)-2-(3-methylphenyl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
2-methyl-1-{2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetyl}-1,4-diazepan-5-one