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1-[(4-methylphenyl)methyl]-4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperazin-2-one
1-[(3,5-difluorophenyl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
4-(benzyloxy)-1-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperidine
7-(4-hydroxy-3-methylbenzoyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-(oxan-4-yl)piperidin-4-ol
methyl[(3-methyloxetan-3-yl)methyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
5-(2-methoxy-4-methylphenoxymethyl)-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide
2-(4-fluorophenyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-1-propyl-1H-pyrazole-5-carboxamide
7-methyl-2-[(2E)-2-methylbut-2-en-1-yl]-2,7-diazaspiro[4.5]decan-6-one
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-5-[1-(4-methylphenyl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazole
1-(azepan-1-yl)-3-[4-chloro-2-({[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)phenoxy]propan-2-ol
4-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
N-[2-(4-hydroxy-3-methoxyphenyl)ethyl]-2-(2,3,6-trimethylphenoxy)acetamide
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-5-[(2,2,3,3-tetrafluoropropoxy)methyl]-1H-1,2,4-triazole
N-[(3S)-1-(3,5-dimethyladamantane-1-carbonyl)pyrrolidin-3-yl]acetamide
1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine-3-carboxamide
(1R,9S)-5-amino-3-(3,5-dimethoxyphenyl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
9-(2-fluoro-2-phenylacetyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{benzyl[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]amino}-2-methylpropan-1-ol
(3R,4R)-3-cyclobutyl-4-methyl-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]pyrrolidin-3-ol
3-(5-methyl-1H-pyrazol-1-yl)-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
N-(propan-2-yl)-1-[(1s,4s)-4-(3,5-dimethoxybenzamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-tert-butyl-3-(2-{[4-(trifluoromethyl)phenyl]carbamoyl}ethyl)piperidine-1-carboxamide
3-methyl-1-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]butan-1-ol
2-(1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)-1H-1,3-benzodiazole
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-2-(2-methoxyphenyl)ethan-1-one
1-(2-{4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
1-cycloheptyl-4-{[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino}pyrrolidin-2-one
6-{[3-(pyrrolidin-1-yl)propyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
8-methyl-3-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-2-(thiophen-2-yl)quinoline
4-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}thieno[2,3-d]pyrimidine
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
4-(4-{[4-(2-aminoethyl)phenyl]methyl}-2-oxopiperazin-1-yl)benzonitrile
(1S,5R)-6-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-(4-benzylpiperazine-1-carbonyl)-N-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3-carboxamide
4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3-dimethylpiperazin-2-one
6-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]pyridazin-3-amine
5,6-dimethyl-2-{2-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
4-[3-(2-chlorophenoxy)azetidin-1-yl]pyridine
3-[(3R,4S)-1-(2-methyl-5-propylpyrimidin-4-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-cyclopentyl-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-[(3-methylthiophen-2-yl)methyl]propanamide
1-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
methyl (1R,3S,3aR,6aS)-3-(4-hydroxyphenyl)-1-(2-methoxy-2-oxoethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
1-[(3-methoxyphenyl)methyl]-4-[2-(thiophen-2-yl)acetyl]piperazin-2-one
4-(2,3-dimethyl-1H-indole-7-carbonyl)-3-(4-fluorophenyl)piperazin-2-one
1-{1-[2-(1H-1,2,4-triazol-5-yl)benzoyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-[(2-fluorophenyl)methyl]-3-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one