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N,1-diethyl-3-(2-methylpropyl)-N-(oxan-2-ylmethyl)-1H-pyrazole-5-carboxamide
2-methylpropyl 3-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxylate
(2R)-2-{[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]amino}-2-phenylethan-1-ol
1-(1-ethylpiperidin-3-yl)-4-[3-(trifluoromethyl)phenyl]piperazine
ethyl 2-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-2-yl}acetate
N,1-diethyl-3,5-dimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-pyrazole-4-carboxamide
5-oxo-1-{4-[2-(piperidin-1-yl)acetamido]phenyl}pyrrolidine-3-carboxylic acid
2-methyl-4-[4-({methyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenyl]butan-2-ol
2-ethyl-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-4-methyl-1,3-oxazole-5-carboxamide
3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-methyl-1-(quinolin-5-ylmethyl)urea
1-{2-[2-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
2-methyl-4-[5-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)thiophen-2-yl]but-3-yn-2-ol
3-(5-{[4-(4-methyl-1H-imidazol-5-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
5-cyclobutanecarbonyl-1'-[(2E)-2-methylbut-2-en-1-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(pyrazine-2-carbonyl)-1,4-diazepan-5-one
(1R,5S)-3-[3-(pyrrolidine-1-carbonyl)benzenesulfonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methoxy-1-(4-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-1-yl)ethan-1-one
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[2-(phenylsulfanyl)ethyl]piperidine
1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
{4-benzyl-1-[1-(1-phenylethyl)-1H-1,2,3,4-tetrazol-5-yl]piperidin-4-yl}methanol
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)(ethyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
2-(5-cyclopropyl-1H-pyrazol-3-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(3S,9aR)-3-[(benzyloxy)methyl]-8-(2-chlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{[7-(5-acetylthiophen-2-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methyl}-2-methoxyacetamide
2-[2-(pyridin-4-yl)ethyl]-9-[(1s,4s)-4-hydroxycyclohexanecarbonyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[1-cyclohexyl-4-(8-methoxyquinolin-2-yl)piperazin-2-yl]ethan-1-ol
4-[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]-N-(propan-2-yl)pyridine-2-carboxamide
1-(2-propyl-1,3-thiazole-4-carbonyl)azetidine-2-carboxylic acid
3-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-(quinolin-6-yl)urea
2-amino-1-{4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}ethan-1-one
N-{1-[7-(cyclohexylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}-5-(methoxymethyl)furan-2-carboxamide
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
4-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-1-ethyl-1,2-dihydropyridin-2-one
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)butanamide
3-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-(trifluoromethyl)benzamide
1-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-[3-(1H-1,2,3-triazol-1-yl)propyl]urea
2-{4-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]butyl}pyridine
2-[3-(pyridin-3-yl)propyl]-4-(trifluoromethyl)pyridine
N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
7-[(2-chlorophenyl)methyl]-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]benzamide
3-(4-chlorobenzoyl)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidine
3-[(2R,3R,6R)-5-[(2-fluoro-4-methylphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
2-ethyl-9-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
1-(2-hydroxybutanoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[3-(1H-imidazol-1-yl)propyl]benzamide
4-{5-[3-(3-methylbutanoyl)piperidine-1-carbonyl]pyridin-2-yl}benzamide