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N-[(1-{[5-(2-cyanophenyl)furan-2-yl]methyl}piperidin-3-yl)methyl]acetamide
1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-(naphthalene-1-carbonyl)piperidine
9-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-3-oxa-9-azaspiro[5.5]undecane
1-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]-3-(3-methylphenoxymethyl)piperidine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-phenoxy-N-{2-[7-(quinolin-7-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}acetamide
3-(3-fluoro-4-methoxyphenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
N2-cyclopropyl-7-(1,2-oxazole-3-carbonyl)-N4-(prop-2-en-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
(3R,4R)-1-(6-ethyl-2-methylquinoline-4-carbonyl)-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
3-{[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
2-[3-(oxan-4-yl)-5-[(phenylformamido)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(hydroxymethyl)piperidin-1-yl]ethan-1-one
9-(3-chloro-4-methoxybenzoyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
(2R,6R)-4-[(1-ethyl-1H-imidazol-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[(3-methylphenyl)methyl]-4-(1H-pyrrole-3-carbonyl)piperazine
dimethyl[1-(3-{1-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1H-imidazol-2-yl}phenyl)ethyl]amine
3-[(1-acetylpiperidin-4-yl)oxy]-N-(cyclohexylmethyl)-4-methoxybenzamide
3-[(3R,4S)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-N,N-dimethylpropane-1-sulfonamide
1-(5-phenyl-1,2,4-oxadiazol-3-yl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
2-[methyl(2-phenylethyl)amino]-N-(pyridin-4-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
2-[5-(quinolin-2-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
N-[(2S)-1-hydroxy-3-(1H-indol-3-yl)propan-2-yl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
6-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidine-1-carbonyl}pyridin-3-ol
2-(2-{[4-(3-fluorophenoxy)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
N-[2-(4-fluorophenyl)ethyl]-N-({2-[3-(hydroxymethyl)piperidin-1-yl]-7-methoxyquinolin-3-yl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
1-{2-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}piperidine-4-carboxamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]pyrrolidin-3-yl]methanol
{7-[5-(pyrrolidin-1-yl)pyridazin-3-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
3-benzyl-8-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(azepane-1-carbonyl)-1-ethyl-N-[2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1R,2R,6S,7S)-N-(1,3-dihydro-2-benzofuran-5-yl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
(3S,4S)-1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-(4-{[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]amino}-6-methylpyrimidin-2-yl)phenol
1-[(1-butylpiperidin-4-yl)methyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
4,4,4-trifluoro-1-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)butan-1-one
4-(benzyloxy)-1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
3-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-[4-(difluoromethoxy)-2-methylphenyl]-3-methylurea
2-(2-hydroxyethyl)-8-(pyrimidin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-{[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-5-methoxypyridin-4-ol
N-benzyl-N-methyl-1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidin-3-amine
1-(3-chlorophenyl)-4-[(3-{2-[1-(furan-3-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl]piperazine
5-(2-fluorophenyl)-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-(1,3-dihydroxypropan-2-yl)-2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
methyl 5-{2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}pentanoate
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(3-ethoxy-4-methoxyphenyl)methyl]amine
1-ethyl-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-1H-pyrazole-4-carboxamide
4,4,4-trifluoro-1-[2-(3-phenylpropyl)morpholin-4-yl]butan-1-one
4-chloro-2-methoxy-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)benzamide
7-chloro-3-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-1-(prop-2-yn-1-yl)-1,2-dihydroquinolin-2-one