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5-(2-chlorophenyl)-N-[(6-hydroxypyrimidin-4-yl)methyl]-2-methylfuran-3-carboxamide
3-{[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-6-methoxy-1,2-dihydroquinolin-2-one
1-methyl-2-{1-[2-(pyridin-2-yl)ethyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
[(3R,4R)-1-(1,3-dimethyl-1H-indole-2-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-[1-(3-chloro-4-hydroxybenzoyl)piperidin-3-yl]-3-phenylpropan-1-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(3-phenyl-1H-1,2,4-triazol-5-yl)acetamide
5-methyl-6-(pyrrolidine-1-carbonyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)thieno[2,3-d]pyrimidin-4-amine
1-[6-(1H-pyrazol-4-yl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
1-{4-[7-chloro-3-({[2-(4-methoxyphenyl)ethyl]amino}methyl)quinolin-2-yl]piperazin-1-yl}ethan-1-one
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2-(3-fluorophenyl)piperidine
1-[1-(6-fluoro-1H-1,3-benzodiazole-2-carbonyl)piperidin-3-yl]pyrrolidin-2-one
3-(4-methoxyphenyl)-5-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}-1H-pyrazole
N-[(2-chloro-6-fluorophenyl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-ethyl-3-methyl-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4R)-N-(1-benzothiophen-2-ylmethyl)-1-benzyl-4-[(4-fluorophenyl)sulfanyl]-N-methylpyrrolidine-2-carboxamide
N-({1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}methyl)-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
{5-[4-(4H-1,2,4-triazol-3-ylmethyl)piperazine-1-carbonyl]furan-2-yl}methanol
1-(4-benzyl-3-ethyl-5-oxo-1,4-diazepane-1-carbonyl)cyclopropane-1-carboxamide
N-{3-[4-(morpholin-4-ylmethyl)phenoxy]propyl}propanamide
5-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-1-(cyclopropylmethyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[5-(3-methyl-1-propyl-1H-pyrazol-4-yl)-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
cyclohexyl(4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
1-cyclopropanecarbonyl-N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]piperidine-4-carboxamide
2-[3-(pyridin-4-yl)-5-[(pyrimidin-2-ylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-[2-(3-methoxyphenyl)ethyl]-6-(1-phenylcyclohexanecarbonyl)-6-azaspiro[2.5]octane-1-carboxamide
6-fluoro-2-oxo-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-dihydroquinoline-4-carboxamide
3-(3-chloro-1,2-oxazol-5-yl)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylpropanamide
1-(3-aminoazepan-1-yl)-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
3-[N-methyl-1-(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazol-4-yl)formamido]propanamide
methyl (2S,4S)-1-methyl-4-(4,5,6,7-tetrahydro-1,3-benzothiazole-2-amido)pyrrolidine-2-carboxylate
methyl 3-(2-methoxyacetamido)-1-[2-(4-methoxyphenyl)ethyl]-5-[(1-methoxypropan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
2-ethoxy-1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
(3S,4S)-4-(dimethylamino)-1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-ol
4-(2,6-dimethylpyridin-3-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrimidin-2-amine
6-chloro-N,N-dimethyl-3-[({2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}amino)methyl]imidazo[1,2-a]pyridine-2-carboxamide
2-{4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
4-{1-[3-(2-phenylethyl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}pyridine
2-(dimethylamino)-N-(2-methoxyethyl)-4-methyl-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
1-(isoquinolin-5-yl)-3-{1-oxaspiro[4.5]decan-3-yl}urea
N-[(3S,4R)-4-(propan-2-yl)-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}pyrrolidin-3-yl]methanesulfonamide
7-[(3-methylphenyl)methyl]-2-[(2-methylpyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-methyl-2-phenyl-N-{[1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methyl}propanamide
4-({[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]carbamoyl}amino)-N-propylbenzamide
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-4-methoxybenzamide
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]quinoline-8-carboxamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
(2R,3R)-3-{methyl[3-(1H-pyrazol-1-yl)propyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5-methyl-N-{3-[(pyridin-3-yl)amino]propyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
(2R)-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyloxolane-2-carboxamide