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4-(propan-2-yl)-6-[3-(pyridin-4-yl)azetidin-1-yl]-2-(trifluoromethyl)pyrimidine
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-(1,2-oxazolidin-2-yl)propanamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidine
3-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2,6-dimethoxypyridine
3-{[2-(furan-2-yl)phenyl]methyl}-9-methoxy-7-oxo-N-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[2-(azepan-1-yl)ethyl]-N-ethyl-3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
(1R,3S)-7-[(2-chloro-4,6-dimethoxyphenyl)methyl]-7-azaspiro[3.5]nonane-1,3-diol
N-(2-methoxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
methyl 4-[2-amino-3-cyano-6-(2-methylbutan-2-yl)pyridin-4-yl]-1H-pyrazole-3-carboxylate
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-(furan-3-ylmethyl)acetamide
N,2-dimethyl-6-(1-methylpiperidin-3-yl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]pyrimidin-4-amine
2-(1-methylpyrrolidin-2-yl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]acetamide
N-methyl-5-{[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl}furan-2-carboxamide
(2S,4S)-4-acetamido-N-ethyl-1-({9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)pyrrolidine-2-carboxamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
3-[5-(1,3,7-trimethyl-1H-indole-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
8-(5-methyl-1,2-oxazole-3-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
(1R,7S)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-4-oxo-3-(pentan-3-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
7-chloro-4-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-(cyclobutylmethyl)-2-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
1-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2,3-dimethoxy-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
N-(3-methoxypropyl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
1-[2-(3-fluorophenyl)-1,3-benzoxazole-5-carbonyl]-2-methyl-1,4-diazepan-5-one
3,5-dimethyl-4-{3-[2-(1-phenylethyl)-1H-imidazol-1-yl]propyl}-1H-pyrazole
N-[3-(morpholin-4-yl)propyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(2S,4S)-4-amino-1-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrrolidine-2-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
1-{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-methylpiperazine
[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
3-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}benzoic acid
N-(6-methylpyridazin-3-yl)-3-[(3-propylmorpholin-4-yl)methyl]benzamide
1-[4-(methylsulfanyl)phenyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}urea
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
3-methyl-1-propyl-N-[3-(pyridin-4-yl)propyl]-1H-pyrazole-4-carboxamide
N-methyl-2-[3-(methylsulfanyl)phenyl]-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
(4aS,8aR)-6-[(4-oxo-4H-chromen-3-yl)methyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
8-[(4-methoxypyridin-2-yl)methyl]-8-azaspiro[4.5]decane-7,9-dione
4-(6-cyclopropylpyrimidin-4-yl)-9-(2-hydroxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]acetamide
4-phenyl-5-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1-[2-(propan-2-ylsulfanyl)ethyl]-1H-imidazole
1-[2-(ethylsulfanyl)ethyl]-3-[(4-fluorophenyl)methyl]-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-[2-(5-methylthiophen-2-yl)ethyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
1-[2-(4-phenoxyphenyl)ethyl]-1H-imidazole
1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
5-({3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]propanamido}methyl)-N-methyl-1,2,4-oxadiazole-3-carboxamide
2-(3,4-dichlorophenyl)-4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]morpholine