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1-ethyl-N-[2-(2-methoxyphenyl)ethyl]-3-(4-methylpiperazine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(2-methoxyphenyl)methyl]-4-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(1-benzylpyrrolidin-3-yl)methyl]-5-(2-fluorophenyl)-1,2,4-triazin-3-amine
4-[2-(dimethylamino)acetamido]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
4-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-7-(3-chlorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{5-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
5-{[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]methyl}-N-propylpyrimidin-2-amine
1-{4-[(4,8-dimethoxynaphthalen-1-yl)methyl]-1,4-diazepan-1-yl}ethan-1-one
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-3-azaspiro[5.5]undecan-9-amine
4-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-(3-methoxyphenyl)-3-methylpiperazin-2-one
(9aS)-N-{3-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxamide
(3S,4R)-N,N-dimethyl-1-(2-methylbenzoyl)-4-(4-methylphenyl)pyrrolidin-3-amine
5-(4-methanesulfonylphenyl)-2,3-dimethylpyrazine
2-{2-[1-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperidin-2-yl]ethyl}pyridine
3-({4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridin-2-amine
4-(2,2-dimethylpropyl)-3-[2-oxo-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]piperazin-2-one
1-[(1,2-dimethyl-1H-indol-3-yl)methyl]-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(oxolan-2-ylmethyl)piperazine
7-{[4-hydroxy-3-methoxy-5-(prop-2-en-1-yl)phenyl]methyl}-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl][2-(2,3-dimethylphenoxy)ethyl]methylamine
(1S,5R)-6-benzyl-3-[3-(methylsulfanyl)propyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(2-chlorophenyl)methyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methylpyrimidin-2-amine
(3aR,6aR)-2-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{1-[5-(4-methoxyphenyl)furan-2-carbonyl]piperidin-3-yl}-5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]pyrimidine
2-(cyclopentylmethyl)-1-(2-methoxyethyl)-6-methyl-N-[3-(morpholin-4-yl)propyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
methyl 2-[butyl(methyl)sulfamoyl]-6-[2-(2-chlorophenyl)acetyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-(azetidin-1-yl)-1-[4-(1H-pyrazol-1-yl)phenyl]piperidine
2-methoxy-6-{[1,2,4]triazolo[4,3-a]quinolin-1-yl}phenol
2-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-1H-indole
5-[(3,4-dimethoxyphenyl)methyl]-5-{3-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
3-acetamido-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylpropanamide
N-[(4-ethoxyphenyl)methyl]-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}cyclopropanamine
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-[(3-methylphenyl)methyl]pyrrolidin-3-yl]methanol
3-[(7-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine
N-({3-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-N-methyloxan-4-amine
4-(2H-1,3-benzodioxol-5-yl)-N-[2-(dimethylamino)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(2-oxoazepan-1-yl)propanamide
1-{2-[3-benzyl-3-(hydroxymethyl)piperidine-1-carbonyl]phenyl}ethan-1-one
5-oxo-N-[2-(pyrazin-2-yl)ethyl]-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl](methyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
N-methyl-2-[4-(pyridin-4-yl)phenyl]acetamide
4-(3-methylpyrazin-2-yl)benzamide
N,6-dimethyl-N-[(3-methyloxetan-3-yl)methyl]-2-(pyridin-3-yl)pyrimidin-4-amine
9-[(2S)-2-(methylamino)propanoyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(3S,4S)-1-{[3-(hydroxymethyl)-2,4,6-trimethylphenyl]methyl}-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
N-(1-hydroxybutan-2-yl)-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
(1H-imidazol-2-ylmethyl)(methyl){[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amine
2-methyl-N-{5-[2-(4-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}oxane-2-carboxamide
N-[3-(azepan-1-yl)-2-hydroxypropyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-[3-(pyridin-3-yl)propyl]piperidine-3-carboxamide