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6-[(diethylamino)methyl]-N-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-cyclopropyl-6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-methylpyrimidin-2-amine
1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
(3aR,6aR)-2-[3-(4-methoxyphenyl)propanoyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
ethyl 1-{[3-(ethoxycarbonyl)-1H-pyrazol-4-yl]methyl}-4-(2-phenoxyethyl)piperidine-4-carboxylate
1-[1-(2,3-dimethylbenzoyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine
N-cyclopentyl-3-[1-(2,3-dimethylphenyl)-1H-1,2,4-triazol-5-yl]propanamide
N-{1-[(6-methylpyridin-2-yl)methyl]azepan-4-yl}-1H-1,2,3-benzotriazole-5-carboxamide
1-(2,2-dimethylpropyl)-N-[3-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
1-({5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,2,4-oxadiazol-3-yl}methyl)-4-methylpiperazine
4-{4-[(2,6-difluorophenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-ol
1-ethyl-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-methylazepane-2-carboxamide
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-3,5-dimethoxybenzamide
5-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}-2-(propan-2-yl)-1,3-benzoxazole
2-[4-(dimethylamino)phenyl]-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
(3aS,6aR)-3-[3-(4-methoxyphenyl)propyl]-5-(2-methylpropanoyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(3S,4S)-4-cyclopropyl-1-[(5-fluoro-2-methoxyphenyl)methyl]pyrrolidine-3-carboxylic acid
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1-benzofuran-3-carboxamide
3-ethyl-1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-(2,2,2-trifluoroethyl)urea
N-[3-(2,6-dimethylphenoxy)propyl]-N-methyl-4-oxo-3,4-dihydroquinazoline-2-carboxamide
N-[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]pyridin-2-amine
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-phenyl-N-{[1-(1H-pyrazole-4-carbonyl)piperidin-3-yl]methyl}methanesulfonamide
4-{1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]pyrrolidin-2-yl}-3,5-dimethyl-1,2-oxazole
4-(1-benzyl-1H-imidazol-2-yl)-N,N-dimethylpiperidine-1-sulfonamide
9-(morpholine-4-carbonyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-tert-butyl-4-{[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]methyl}furan-2-carboxamide
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}pyridin-2-amine
3-(methoxymethyl)-1-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidine
4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]-N,N-dimethylpiperidine-1-sulfonamide
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4-diazepan-6-yl]oxy}acetamide
4-(1-phenyl-1H-pyrazol-4-yl)-2-[4-(pyrazin-2-yl)piperazin-1-yl]pyrimidine
1-{2-oxo-2-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[4-(benzyloxy)piperidin-1-yl]-3-[methyl(1-methylpyrrolidin-3-yl)amino]propan-1-one
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)oxane-4-carboxamide
methyl 4-({2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxyphenyl}formamido)butanoate
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[4-(1H-pyrazol-1-yl)butan-2-yl]propanamide
2-(4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl)ethan-1-ol
N,N-dimethyl-5-{[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]methyl}pyridin-2-amine
2-ethoxy-1-{4-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethan-1-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-4,4,4-trifluorobutanamide
4-chloro-1-ethyl-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-1H-pyrazole-5-carboxamide
3-(4-chloro-1H-pyrazol-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
1-(3-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-3-oxopropyl)pyrrolidin-2-one
4-{3-[4-(1-methylpiperidin-4-yl)piperazine-1-carbonyl]phenyl}morpholine
3-{[ethyl(2-methylprop-2-en-1-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-{3-[4-({[3-(trifluoromethoxy)phenyl]methyl}amino)piperidin-1-yl]phenyl}cyclopropanecarboxamide