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(1S,5R)-3-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-chlorophenyl)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetamide
[1-(2-{[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}ethyl)piperidin-2-yl]methanol
1-tert-butyl-4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
2-ethyl-5-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]pyrimidine
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(4-methylpyridin-2-yl)pyrrolidine-3-carboxylic acid
N-(4-chloro-3-methylphenyl)-2-[4-(cyclopropylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]acetamide
N-[1-(2-phenylethyl)piperidin-3-yl]-5-propyl-1,2-oxazole-4-carboxamide
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-5-(5-methylfuran-2-yl)-1,2,4-triazin-3-amine
7-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-chloro-N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-(2-methoxy-6-methylphenyl)benzamide
N,1,5,6-tetramethyl-2-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2-dihydropyridine-3-carboxamide
3-hydroxy-3-({[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
N-[3-(1H-indazol-1-yl)propyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
1-{3-[4-phenyl-5-(pyridin-4-yl)-1H-imidazol-1-yl]propyl}pyrrolidin-2-one
N'1-[2-(dimethylamino)ethyl]-N'1-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)cyclopropane-1,1-dicarboxamide
5-{[4-(2-methoxyethoxy)piperidin-1-yl]methyl}-1-methyl-1H-indole
4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1-methyl-1H-indole
2-({[(3R,4R)-1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
(3aS,6aS)-2-[(2-chloro-4-fluorophenyl)methyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-fluoro-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-(morpholin-4-yl)pyrimidin-2-amine
N-(1,2-oxazol-3-ylmethyl)-5-(oxolan-2-yl)thiophene-2-carboxamide
1-{4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}piperidin-3-ol
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
4-(2-methyl-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-2-yl)morpholine
4-{[4-(4-methylphenyl)-4H-1,2,4-triazol-3-yl]methyl}pyridine
3-[4-(2-methoxyphenyl)-1,3-dimethyl-1H-pyrazol-5-yl]-1-[1-(1-methyl-1H-pyrazol-5-yl)propyl]urea
6-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyrrolidin-1-yl)pyrimidin-4-amine
2-(5-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}thiophen-2-yl)-1H-imidazole
6-chloro-N,1-dimethyl-N-[1-(pyridin-3-yl)pentyl]-1H-indole-2-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}propanamide
5-ethyl-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
(3S,9aR)-3-ethyl-8-[(2-fluoro-5-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(pyridin-2-ylmethyl)-4-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
N-benzyl-4-cyano-4-phenylpiperidine-1-sulfonamide
6-ethoxy-3-({methyl[(1-methylpyrrolidin-3-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-amino-4-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
3-{methyl[1-(methylcarbamoyl)ethyl]sulfamoyl}-N-[3-(methylsulfanyl)propyl]benzamide
2-(4-chlorophenyl)-4-[5-(morpholine-4-carbonyl)pyridin-2-yl]morpholine
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-N-(cyclohexylmethyl)propanamide
2-{3-[3-(3-cyanopyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}-N-(1,3-thiazol-2-yl)propanamide
N-(1-{1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
5,7-dimethyl-2-[2-(propan-2-yl)pyrimidin-5-yl]-4-(pyrrolidine-1-carbonyl)quinoline
2-methyl-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
ethyl 3-({3-[4-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}amino)propanoate
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide