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N-methyl-5-(4-methylphenyl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1H-pyrazole-3-carboxamide
1-[3-(azepane-1-carbonyl)phenyl]-3-[(1R)-2,3-dihydro-1H-inden-1-yl]urea
1-[4-(6-methyl-9H-purin-9-yl)phenyl]ethan-1-ol
2-[1-(butan-2-yl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-6-methylpyridine
N-ethyl-8-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-1-methyl-N-(pyridin-4-ylmethyl)piperidin-4-amine
2-{2-[(6-hydroxy-1,4-oxazepan-4-yl)methyl]phenoxy}-1-(4-methylpiperidin-1-yl)ethan-1-one
1-{[(3R,4R)-1-[4-(dimethylamino)benzoyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
1-(1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-4-yl)pyrrolidin-2-one
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N,5,7-trimethylpyrido[2,3-d]pyrimidin-4-amine
3-(2-methyl-1H-imidazol-1-yl)-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)propanamide
1-(azocan-1-yl)-3-(2-methoxy-4-{[(1-methylpiperidin-4-yl)amino]methyl}phenoxy)propan-2-ol
5-cyclopentyl-3-{[5-(1-ethyl-1H-1,2,4-triazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
{1-[2-({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)ethyl]piperidin-3-yl}methanol
1-methyl-4-(pyrrolidine-1-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1'-[4-(furan-2-yl)benzoyl]-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-amino-3-ethyl-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-phenyl-3-(piperidin-3-yl)-1-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(morpholin-4-yl)-1-{4-[2-(pyridin-3-yl)-1H-imidazol-1-yl]phenyl}ethan-1-ol
9-[(4-ethenylphenyl)methyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
(5S,9aS,9bS)-5-(3-chloro-4-hydroxyphenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-(pyridin-2-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-2-amine
1-ethyl-5-{[(3-phenyl-1H-pyrazol-5-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[(2S)-1-hydroxypropan-2-yl]-2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
2-amino-6-ethyl-4-[2-(ethylsulfanyl)pyrimidin-5-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-(cyclohex-1-en-1-ylmethyl)-1-(furan-2-ylmethyl)piperidine-3-carboxamide
(2S)-2-hydroxy-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-3-phenylpropanamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-1H-indole-6-carboxamide
N-[1-(1H-1,2,4-triazol-5-yl)ethyl]-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
9-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylpyridine-3-carboxamide
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N-(2-methylpropyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}piperidine-3-carboxamide
[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl][(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]methylamine
(3S,5S)-1-(2-methoxy-2-methylpropanoyl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
2-(6-methyl-1-benzofuran-3-yl)-N-[2-(1-methylpiperidin-3-yl)ethyl]acetamide
N-cyclopropyl-1-methyl-5-phenyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrrole-2-carboxamide
4-{7-[2-(ethylsulfanyl)propanoyl]-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}benzamide
4-methoxy-N-[2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]benzene-1-sulfonamide
2-(2-methoxyethyl)-8-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(1-phenylbutyl)propanamide
[4-({methyl[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)oxan-4-yl]methanol
7-[2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)acetyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-ethyl-3-(piperidine-1-carbonyl)-N-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{1-[(cyclopropylcarbamoyl)methyl]piperidin-4-yl}-4-(4H-1,2,4-triazol-4-yl)benzamide
(3S,4R)-4-(3-fluorophenyl)-1-(oxane-4-carbonyl)pyrrolidine-3-carboxylic acid
1-methyl-4-({5-[1-(1H-pyrazol-1-yl)propan-2-yl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
(1S,5R)-3-methyl-6-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N4-{[1-(dimethylamino)cyclohexyl]methyl}-6-methylpyrimidine-2,4-diamine
1-(2-amino-4-phenylpyrimidine-5-carbonyl)azepan-4-amine
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione