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N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-amine
2-{3-[(3-methylpiperidin-1-yl)methyl]phenyl}-6-(3-methylpyrazin-2-yl)-3,4-dihydropyrimidin-4-one
3-hydroxy-3-({[2-(piperazin-1-yl)ethyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
1-(2,3-dihydro-1H-inden-2-yl)-5-[1-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-1,2,4-triazole
1-methyl-2-oxo-8-[2-(pyridin-2-yl)ethyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N,5-dimethyl-N-(2-methylpropyl)-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
3-(3-hydroxy-1,2-oxazol-5-yl)-1-{2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}propan-1-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-cyclohexanecarbonyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyridine-3-sulfonamide
4-(2,4-difluorophenyl)-3-(4-hydroxy-3-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[4-(1-benzofuran-2-yl)phenyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-[7-(3-chlorophenyl)-9-(furan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenylethan-1-one
1-(2-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}-2-oxoethyl)-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2R,6R)-4-(2,5-dimethylbenzoyl)-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(3R,5R)-N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-4-(4H-1,2,4-triazol-4-yl)benzamide
4-{[1-(3-chlorophenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}morpholin-2-one
2-{2-[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
N-(4-butanamido-3-methoxyphenyl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
5-fluoro-N2-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-N4,N4-dimethylpyrimidine-2,4-diamine
N-{[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-3-yl]methyl}-1-(4-chlorophenyl)cyclopropane-1-carboxamide
2-methoxy-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
methyl 6-{[(2-methoxyethyl)(propan-2-yl)amino]methyl}-3-(4-methylbenzamido)thieno[2,3-b]pyridine-2-carboxylate
3-[(1-benzothiophen-2-ylmethyl)amino]-N-(4-methoxyphenyl)-5-(methylsulfamoyl)benzamide
3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propyl-5-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
N-methyl-2-(4-methylpiperazine-1-carbonyl)-N-(2-phenylethyl)-2,3-dihydro-1H-inden-2-amine
N-{1-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
methyl 5-[2-(4-chlorophenyl)morpholin-4-yl]pentanoate
N-[3-(4-chlorophenoxy)-2-hydroxypropyl]-2-(ethylamino)pyrimidine-5-carboxamide
1-{4-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
7-methyl-2-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-cyclopropylquinoline-4-carboxamide
methyl (2S)-1-[2-(2-methoxyphenoxy)ethyl]pyrrolidine-2-carboxylate
7-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-(2-methylpyridin-4-yl)-4-(oxolan-3-ylmethyl)-1,4-diazepane
N-(3-hydroxy-2,2-dimethylpropyl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
ethyl 4-[3-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)propanoyl]piperazine-1-carboxylate
5-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1,3-benzothiazol-2-amine
1-[4-(adamantan-1-yl)piperazin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-methyl-3-(1-methylpiperidin-2-yl)-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}propanamide
1-{1-[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
methyl 1-methoxy-2-oxo-8-[1-(pyridin-2-yl)piperidine-3-carbonyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[3-(methylsulfanyl)propanoyl]-decahydro-1,6-naphthyridin-2-one
N-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}-N-methyloxan-4-amine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[(1R)-2,2,2-trifluoro-1-phenylethyl]propanamide
N-(1-{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}pyrrolidin-3-yl)acetamide