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5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(4-methylpiperazin-1-yl)ethyl]piperidin-2-one
7-[2-(morpholin-4-yl)propanoyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2R,3R)-1'-(6-chloropyridazin-3-yl)-3-[ethyl(methyl)amino]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-[2-(2-fluorophenyl)ethyl]-3-(3-methoxypropyl)-3-(1-methylpiperidin-4-yl)urea
methyl 1-ethoxy-8-(9H-fluoren-2-ylmethyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-(1-methyl-1H-pyrazol-5-yl)-2-{4-[5-(piperazin-1-ylmethyl)thiophen-3-yl]-1H-pyrazol-1-yl}acetamide
4-methoxy-2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
1-[(3-methoxyphenyl)methyl]-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
1-(2-methylphenyl)-4-[3-(2-oxopyrrolidin-1-yl)propanoyl]piperazin-2-one
4-[5-(3-methylfuran-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]morpholine
3-(3-methoxypropyl)-1-(3-methylpyrazin-2-yl)piperidine-3-carboxylic acid
2-(3-methyl-1H-pyrazol-1-yl)-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]acetamide
3-[1-(5-hydroxypyrazine-2-carbonyl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
N-[(2S)-1-methoxypropan-2-yl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
3-[(4-acetylmorpholin-2-yl)methyl]-1-[4-(2-fluorophenoxy)phenyl]urea
3-cyclopropyl-1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
1-[(2-chloro-6-fluorophenyl)methyl]-5-(1,3-thiazol-4-ylmethyl)-1H-1,2,4-triazole
5-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
(2Z)-1-[(4aR,8aS)-6-(5-acetylthiophene-3-carbonyl)-decahydro-1,6-naphthyridin-1-yl]-2-fluoro-3-phenylprop-2-en-1-one
8-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
N-cyclohexyl-4-(4-methyl-1,2,3-thiadiazole-5-amido)piperidine-1-carboxamide
4-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-6-(morpholin-4-yl)pyrimidin-2-amine
({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)(1,3-thiazol-5-ylmethyl)amine
2-[1-(6-methoxy-3-methyl-1-benzofuran-2-yl)-N-methylformamido]-2-(thiophen-2-yl)acetic acid
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-(methylsulfanyl)propanamide
4-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
(S)-(2-chlorophenyl)[1-(4-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methanamine
N-[(3S,4R)-1-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
methyl 4-[({1-[(3-methoxyphenyl)methyl]piperidin-3-yl}amino)methyl]benzoate
(2E)-N-({7-[3-(1H-indol-3-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenylprop-2-enamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-1-(3-cyclohexylpyrrolidin-1-yl)propan-1-one
N-methyl-4-({2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)-1,3-thiazol-2-amine
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-(pyrrolidin-3-yl)benzamide
1-benzyl-N-(butan-2-yl)-5-methyl-N-(3-phenylprop-2-yn-1-yl)-1H-1,2,3-triazole-4-carboxamide
3-chloro-N-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzamide
N-[(5-chloro-2-methoxyphenyl)methyl]-3-fluoro-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
2,2-dimethyl-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}thiomorpholin-3-one
N-(3-cyclopentylpropyl)-1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carboxamide
4-(2-phenylethyl)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-3-phenylpropanamide
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]propanamide
1-[4-(morpholin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-3-(1H-pyrazol-1-yl)propan-1-one
(4S)-3,3,4-trimethyl-1-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-ol
3-(2H-1,3-benzodioxol-5-yl)-N-[(5-methylpyrazin-2-yl)methyl]-3-phenylpropanamide
6-(benzyloxy)-4-(oxolane-3-carbonyl)-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
N,N-dimethyl-2-[(1S,5R)-6-[2-(pyrrolidin-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
1-methyl-N-[3-(morpholin-4-yl)propyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
3-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-N-(furan-2-ylmethyl)propanamide
1-[1'-(2-ethylpyridine-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
7-(1H-1,2,3-benzotriazole-5-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one