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3-ethoxy-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}propan-1-one
1-[1-(5-chloro-2-methylpyrimidine-4-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-methyl-1H-pyrazole-5-carboxamide
ethyl 4-benzyl-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylate
4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-(3-ethoxypropyl)pyridine-2-carboxamide
[1-(furan-3-carbonyl)-3-(3-phenylpropyl)piperidin-3-yl]methanol
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidine
N-[(2S,4R,6S)-2-benzyl-6-{6-methylimidazo[2,1-b][1,3]thiazol-5-yl}oxan-4-yl]acetamide
4-(benzylsulfamoyl)-N-(oxolan-3-yl)benzamide
4-(2-{4-[3-(1H-pyrrol-1-yl)propanoyl]morpholin-3-yl}acetyl)piperazin-2-one
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-[2-(1H-indol-3-yl)ethyl]acetamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
1-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-4-(2-methoxyethyl)piperazine
1-[2-({5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}amino)ethyl]piperidin-4-ol
N-[3-(4-hydroxyphenyl)propyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
7-{[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl}-2,7-diazaspiro[4.5]decane
2-[2-(cycloheptylamino)pyrimidin-4-yl]pyridine-4-carboxylic acid
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(2,6-dimethylpyrimidine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-amino-7-(4-methyl-5-phenylthiophene-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-2-(morpholin-2-yl)acetamide
2-(4,6-dimethyl-1-benzofuran-3-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]ethan-1-one
methyl[(1-methyl-1H-imidazol-2-yl)methyl]{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
7-(3-chlorophenyl)-4-(1-methyl-1H-pyrrole-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-5-propyl-1,2-oxazole
3-[1-(2-acetamidoacetyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
2-(dimethyl-1,3-thiazol-5-yl)-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]acetamide
propan-2-yl 4-chloro-3-[2-(1H-imidazol-2-yl)benzamido]benzoate
5-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}imidazo[1,2-a]pyridine-2-carboxamide
4-{[5-(1-benzyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-methylpiperidine
N-(4-methoxy-2-methylphenyl)-3-[1-(thian-4-yl)piperidin-3-yl]propanamide
2-(4-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-ol
methyl (2S)-1-[4-(cyclopropylamino)-5-methylthieno[2,3-d]pyrimidine-6-carbonyl]pyrrolidine-2-carboxylate
1-{4-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one
2-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]methyl}-1H-imidazole
3-(methoxymethyl)-5-[(E)-2-[4-(trifluoromethyl)phenyl]ethenyl]-1H-1,2,4-triazole
6-{[(dimethylcarbamoyl)methyl]amino}-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
2-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-4-(1H-pyrrol-1-yl)phenol
2,6-dimethoxy-N-[1-(3-phenylpropyl)piperidin-3-yl]benzamide
2-(2-chloro-4-fluorophenyl)pyridine-4-carboxamide
{[4-methoxy-3-(methoxymethyl)phenyl]methyl}(methyl)(thiophen-3-ylmethyl)amine
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(3-hydroxypiperidin-1-yl)ethan-1-one
6-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
N-[(3S,5S)-1-(cyclobutylmethyl)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
(1R,7S)-N-(furan-3-ylmethyl)-3-[4-(2-hydroxyethyl)phenyl]-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-{[1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]methyl}naphthalene-1-carboxamide
8-(1-phenylcyclopentanecarbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(2-chlorophenyl)methyl 1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxylate
methyl 4-[4-(5-hydroxypyrazine-2-carbonyl)piperazin-1-yl]benzoate