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1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3,3-diphenylpiperidine
2-methyl-3-{[2-(pyridin-3-yl)morpholin-4-yl]methyl}quinoxaline
4-(4-cyclopentyl-1,4-diazepane-1-carbonyl)-2-fluorophenol
3-(2-fluorophenyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
2-(dimethyl-1,3-thiazol-5-yl)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
2-[4-(3,5-difluorophenyl)phenoxy]-N-methylacetamide
2-(3-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}piperidin-1-yl)acetamide
methyl[1-(pyrazin-2-yl)propan-2-yl](4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-5-phenylpentan-1-one
2-[4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)morpholin-2-yl]ethan-1-amine
(2E)-N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)-3-(thiophen-2-yl)prop-2-enamide
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
3-methyl-4-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]benzoic acid
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-oxo-2-phenylacetamide
3-[2-methyl-3-(pyrrolidine-1-carbonyl)phenyl]-1-(oxan-4-yl)urea
[(2S,4R)-4-(dimethylamino)-1-(2,2-diphenylethyl)pyrrolidin-2-yl]methanol
(4aS,7aR)-1-(5-methyl-1,3-oxazole-4-carbonyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(1,2-oxazinan-2-yl)-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propan-1-one
(2S,4R)-4-amino-1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-N-methylpyrrolidine-2-carboxamide
1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-2-(pyridin-2-ylsulfanyl)ethan-1-one
(2S)-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]piperidine-2-carboxamide
N-methyl-3-(N-methylmethanesulfonamido)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}propanamide
(4aS,7aR)-1-[2-(azepan-1-yl)-2-oxoethyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,4R)-4-methyl-3-(propan-2-yl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]pyrrolidin-3-ol
(3R,4R)-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-2-methyl-1H-1,3-benzodiazole
2,2-diphenyl-1-[4-(thiophene-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]ethan-1-ol
5-(1-benzothiophen-2-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N1,N1-dimethyl-N3-[3-(3-methylphenyl)propyl]piperidine-1,3-dicarboxamide
1-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]azepane
8-[2-(propan-2-yloxy)acetyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
[(3R,4R)-1-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(4-methoxyphenyl)acetamide
3-[1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-(2-ethoxyphenyl)-N-(1-ethyl-1H-1,2,4-triazol-3-yl)piperazine-1-carboxamide
1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-1-methyl-N,3-dipropyl-1H-pyrazole-5-carboxamide
2-[4-(3-fluorophenoxy)piperidine-1-carbonyl]-N,N-dimethylaniline
2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)-N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
4-phenoxy-1-[2-(pyrrolidin-1-yl)acetyl]piperidine-4-carboxylic acid
3-methyl-7-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-(1H-imidazol-1-ylmethyl)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-4-ol
N-tert-butyl-6-methyl-5-[5-(pyridin-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
3-(5-methoxy-2-methylphenyl)-1-(oxan-4-yl)urea
(4S,4aS,8aS)-1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-phenyl-decahydroquinolin-4-ol
N-methyl-5-[2-(2,5,7-trimethyl-1H-indol-3-yl)acetyl]-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(4-chlorophenyl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]butanamide
N-{[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-3-yl]methyl}-1-(4-chlorophenyl)cyclopropane-1-carboxamide
(1R,3S)-3-(2-aminoethoxy)-7-[2-(ethylamino)pyrimidine-5-carbonyl]-7-azaspiro[3.5]nonan-1-ol