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methyl[(8-methylquinolin-5-yl)methyl][3-(oxolan-2-yl)propyl]amine
N-(1-benzylpiperidin-4-yl)-6-methoxypyrimidin-4-amine
4-({3-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)-1,4-diazepane-1-carbaldehyde
3-(2-ethyl-1H-imidazol-1-yl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylpropanamide
6-(4-methoxyphenyl)-7-methyl-2-(2-methylpyrrolidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
3-benzyl-1-(2-phenylethyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-chloro-4-fluoro-N-[2-(methylsulfamoyl)ethyl]-1-benzothiophene-2-carboxamide
1-[3-(4-{[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one
2-methoxy-3-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
3-{5-[2-(3-phenylpyrrolidin-1-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
ethyl 1-[(4-hydroxyquinolin-2-yl)methyl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
5-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
2-{[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]methyl}-6-methylpyridin-3-ol
(3S,4S)-1-(2-methoxypyrimidine-5-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
4-(2,6-dimethoxybenzoyl)-1-phenylpiperazin-2-one
(3aR,6aR)-2-methanesulfonyl-5-[(1-methyl-1H-indol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(2-methylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1-methyl-1H-indole-2-carboxamide
6-(propan-2-yloxy)-N4-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}pyrimidine-2,4-diamine
(3R,5S)-5-[1-cyclohexyl-3-(3-methoxyphenoxymethyl)-1H-1,2,4-triazol-5-yl]pyrrolidin-3-ol
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}propanamide
1-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
4-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
4-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(1R,7S)-3-cycloheptyl-N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
5-[(2-methylphenyl)methyl]-5-(piperidin-4-yl)-3-[2-(pyridin-4-yl)ethyl]imidazolidine-2,4-dione
5-(2-chlorophenyl)-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methylfuran-2-carboxamide
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-6-methoxyhexan-1-one
1-(2-methoxyethyl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-6-oxopiperidine-3-carboxamide
2-[(3-chloro-1-benzothiophen-2-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-(1-{1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
3-[1-(5-phenoxyfuran-2-carbonyl)azetidin-3-yl]pyridine
3,3-diethyl-1-{4-[3-(methylsulfanyl)-1H-1,2,4-triazol-5-yl]phenyl}urea
[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl){[3-(pyrimidin-2-yloxy)phenyl]methyl}amine
N-(butan-2-yl)-6-(2-fluoro-4-methoxyphenyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-4-(1H-1,2,4-triazol-1-yl)butanamide
3,5-dimethyl-7-[3-(5-methylfuran-2-yl)benzoyl]-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N,N-diethyl-1H-pyrazole-4-carboxamide
6-methyl-5-{5-[3-(5-methylthiophen-2-yl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
(1S,5R)-3-(4-fluoro-3-methylbenzoyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
8-[2-(ethylamino)pyrimidine-5-carbonyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-4-yl}pyrrolidine-1-carboxamide
3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-N-(6-methylpyridin-3-yl)benzamide
3-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-1-(4-methylpiperazin-1-yl)propan-1-one
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-4-methoxybenzamide
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-3-carboxamide
3-methyl-4-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-1-(2-methylpropyl)piperazin-2-one
6-methyl-5-[5-(1,2,3,4-tetrahydronaphthalen-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
5-(2,4-dimethoxyphenyl)-N-[2-(2-fluorophenyl)ethyl]-1,2,4-triazin-3-amine