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N-[(3S,4R)-4-(4-methylphenyl)-1-(9H-purin-6-yl)pyrrolidin-3-yl]cyclopropanecarboxamide
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-3-(1H-pyrazol-4-yl)propanamide
2-(dipropylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
8-[(9-ethyl-9H-carbazol-3-yl)methyl]-1-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N,N-diethyl-2-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}acetamide
2-butyl-N-methyl-N-(oxolan-3-yl)-1,3-benzoxazole-5-carboxamide
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1-propyl-1H-pyrazole-5-carboxamide
3-{2-[4-(2-hydroxyethyl)piperazin-1-yl]-4-(4-methylphenyl)pyrimidin-5-yl}benzonitrile
N-{2-[({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]ethyl}pyridine-4-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-[(4-methoxyphenyl)methyl]-N-(oxolan-2-ylmethyl)acetamide
7-(4-propylbenzoyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[4-(3-fluoro-2-methoxybenzoyl)-1-(furan-2-ylmethyl)piperazin-2-yl]ethan-1-ol
2-ethyl-9-methanesulfonyl-4-phenyl-2,9-diazaspiro[5.5]undecane
1-cyclopropanecarbonyl-4-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}piperidine
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N,1-dimethyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{2-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}azonan-2-one
1-cyclopentyl-4-[2-methoxy-4-(3-methoxypiperidine-1-carbonyl)phenoxy]piperidine
N-[3-({[1-(3-chlorophenyl)cyclopropyl]carbamoyl}amino)-2-methylphenyl]-2-methoxyacetamide
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(3-ethoxy-2-hydroxypropyl)amine
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]pyrazine-2-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-5-(propan-2-yl)pyrimidin-4-amine
2,6-dimethoxy-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyridine-3-carboxamide
N,2-dimethyl-N-[3-(1H-pyrazol-1-yl)propyl]thieno[3,2-d]pyrimidin-4-amine
2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-1-(prop-2-en-1-yl)-1H-1,3-benzodiazole
(3aS,6aR)-N-tert-butyl-3-[(3,4-dimethoxyphenyl)methyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]acetamide
5-[bis(prop-2-en-1-yl)amino]-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[4-(ethanesulfonyl)morpholin-3-yl]-1-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethan-1-one
(4aS,7aR)-1-(4-methyl-1H-pyrrole-2-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-hydroxy-N-[2-(5-methylthiophen-2-yl)ethyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-[5-(hydroxymethyl)furan-2-carbonyl]piperazin-2-one
2-(pyrimidin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-methyl-6-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridazine
N,N-dimethyl-4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine-1-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}propanamide
4-(2,6-dimethylpyridin-4-yl)-N-(1H-indazol-7-yl)piperazine-1-carboxamide
1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-(2-methylpropyl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-5-phenyl-1,2-oxazole-3-carboxamide
5-(2,5-dimethylphenoxymethyl)-N-methyl-N-(quinolin-2-ylmethyl)-1,2-oxazole-3-carboxamide
6-[4-(2-phenoxyethyl)piperazine-1-carbonyl]piperazin-2-one
(2S)-2-[2-(3-methyl-1-benzofuran-2-yl)-1H-imidazol-1-yl]-4-(methylsulfanyl)butan-1-ol
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
5-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-N-(propan-2-yl)pyrimidin-2-amine
(1S,5R)-3-benzyl-6-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N'-(2-ethoxyphenyl)-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]propanediamide
4-methyl-N-({1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)-1,2,3-thiadiazole-5-carboxamide
3-{[(2-methoxyethyl)[(5-methylthiophen-2-yl)methyl]amino]methyl}pyrrolidin-3-ol
5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-[(4-methoxyphenyl)methyl]-1H-pyrazole-4-carboxamide