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N-[(1-ethylpyrrolidin-2-yl)methyl]-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
(3R,4R)-1-(6-methyl-2-phenylpyrimidin-4-yl)-4-(morpholin-4-yl)piperidin-3-ol
N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-1-phenylcyclohexane-1-carboxamide
(5S,9aS,9bS)-5-[(E)-2-(furan-2-yl)ethenyl]-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2,4-dimethyl-N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-1,3-thiazole-5-carboxamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
8-(1H-indol-5-ylmethyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
5-(3,4-dimethylphenoxymethyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-N,2-dimethyl-2-(1H-pyrrol-1-yl)propanamide
1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(3S,4S)-1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-6-(indolizin-2-yl)pyridine-3-carbonitrile
5-({[3-(thiophen-3-yl)-1,2,4-oxadiazol-5-yl]methyl}sulfanyl)-1,3,4-thiadiazol-2-amine
N-ethyl-4-(2-propyl-1,3-thiazole-4-amido)piperidine-1-carboxamide
8-(cyclohex-3-en-1-ylmethyl)-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
N-(1-{1-[1-(3-methylphenyl)piperidin-4-yl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
3-[2-oxo-2-(3-propylmorpholin-4-yl)ethyl]-2,3-dihydro-1,3-benzoxazol-2-one
N-(2-{4-[(2-methylphenyl)methyl]morpholin-2-yl}ethyl)-1,3-oxazole-5-carboxamide
1-tert-butyl-3-(furan-2-yl)-5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-1,2,4-triazole
N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)oxolane-2-carboxamide
(3R,4S)-1-(1-benzofuran-5-carbonyl)-4-cyclopropylpyrrolidin-3-amine
4-{3-[(5-methoxy-1-methyl-1H-indol-2-yl)formamido]propyl}-1,2,5-oxadiazole-3-carboxylic acid
1-(4-chloro-1-ethyl-1H-pyrazole-3-carbonyl)-4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]ethan-1-one
(2S,4S)-4-amino-N-methyl-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidine-2-carboxamide
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-(4-fluorobenzenesulfonyl)-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(1,2,4-oxadiazol-3-ylmethyl)-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
3-(5-methyl-2,1,3-benzothiadiazol-4-yl)-1-[3-(3-oxopiperazin-1-yl)propyl]urea
2-ethoxy-1-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethan-1-one
4-{1-benzyl-5-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
2-[1-(cyclohexylmethyl)-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl]ethan-1-ol
(3S,4S)-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine-3,4-diol
3-[1-(thian-4-yl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)acetamide
4-{[3-hydroxy-2-oxo-1-(3-phenylpropyl)piperidin-3-yl]methyl}piperazin-2-one
1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
3-({4-[3-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)-1λ6-thiolane-1,1-dione
3-methyl-2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]pyridine
(2R,3R)-3-amino-1'-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[(5-methylthiophen-2-yl)methyl]-5-(propan-2-yl)-N-(pyridin-2-ylmethyl)-1,2-oxazole-3-carboxamide
(1R,2R,6S,7S)-N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
1-[3-methyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-6-azaspiro[2.5]octane
4-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-(2-oxo-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}ethyl)piperazin-2-one
1-[(2-fluorophenyl)methyl]-6-oxo-N-(pentan-3-yl)piperidine-3-carboxamide
methyl 2-[3-oxo-4-(pyrimidin-2-ylmethyl)-3,4-dihydro-2H-1,4-benzoxazin-2-yl]acetate
1-(2-methoxyethyl)-3-[1-(2-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]piperidine
N-cyclopropyl-2-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyridine-4-carboxamide
N-[(2,5-dichlorophenyl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-[(2,4,5-trimethylphenyl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-N-(oxolan-2-ylmethyl)thiophene-2-sulfonamide