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3-phenyl-1-[4-(3-phenyl-1H-pyrazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]propan-1-ol
N-methyl-N-[3-(morpholin-4-yl)propyl]-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
2-({4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
N4-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N4-methyl-2-(pyrrolidin-1-yl)pyrimidine-4,6-diamine
6-ethyl-1,5-dimethyl-3-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
N-[(2-methoxyphenyl)methyl]-4-(4-methylphenoxy)piperidine-4-carboxamide
methyl 4-({2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}amino)benzoate
N-(3-ethoxypropyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-2-(pyridine-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline
3-[(2R,3R,6R)-5-cyclobutanecarbonyl-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
2-tert-butyl-N-[1-(2-fluorophenyl)piperidin-4-yl]-4-hydroxypyrimidine-5-carboxamide
4-(3-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(carbamoylmethyl)-N-methylpropanamide
2-[3-(2-methoxyphenoxy)azetidin-1-yl]-4-(pyrrolidine-1-carbonyl)pyridine
6-methyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
6-({2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-3-ethyl-3H-imidazo[4,5-b]pyridin-2-amine
3-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
1-methyl-4-({2-[4-(pyrimidin-2-yloxy)phenyl]-1H-imidazol-1-yl}methyl)piperidin-4-ol
1-(2,3-dihydro-1H-inden-2-yl)-4-({[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}amino)pyrrolidin-2-one
2-(2-chloro-6-fluorophenyl)-N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-methylacetamide
(2S,4S)-4-amino-N-(propan-2-yl)-1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidine-2-carboxamide
4-[1-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-1H-imidazol-2-yl]quinoline
N-[4-methyl-3-(2-oxopyrrolidin-1-yl)phenyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-methanesulfonyl-N-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-amine
1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-2-[(2-methylphenyl)sulfanyl]ethan-1-one
(3R,9aR)-3-benzyl-8-(3-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-(2-methylphenoxy)-1-[2-(pyridin-3-yl)acetyl]piperidine-4-carboxylic acid
N-(dimethyl-1H-1,2,4-triazol-5-yl)-5-[1-(oxan-4-ylmethyl)pyrrolidin-2-yl]thiophene-2-carboxamide
[(3R,4R)-1-(2-chlorobenzoyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
2-[2-(ethylsulfanyl)ethyl]-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}-3-(1-methylpiperidin-3-yl)propanamide
[2-ethoxy-5-({3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenyl]methanol
dimethyl(2-{4-[2-(5-methylfuran-2-yl)phenyl]-1H-1,2,3-triazol-1-yl}propyl)amine
5-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-N-ethylpyrimidin-2-amine
1-methyl-9-[3-(1H-pyrazol-4-yl)benzoyl]-1,4,9-triazaspiro[5.5]undecan-5-one
1-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
2-(1H-imidazol-2-yl)-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)benzamide
3-methyl-4-(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,2,5-oxadiazole
1-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-4-methylpentane-1,2-dione
2-(benzylsulfanyl)-5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}pyrimidine
1,3-dimethyl-5-(2-oxo-2-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazin-1-yl}ethyl)imidazolidine-2,4-dione
2-(1-{[1-(1-ethyl-3-methylpiperidine-3-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]methylamine
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[(2S)-1-hydroxybutan-2-yl]pyrimidine-5-carboxamide
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](ethyl){[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}amine
3-(dimethyl-1,2-oxazol-4-yl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
1-methyl-N-{2-[2-(3-methylbutoxy)phenyl]ethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
6-{[(6-hydroxypyrimidin-4-yl)methyl]amino}-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
7-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine