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1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(thiophene-2-carbonyl)piperidine
N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)-2-(1H-1,2,4-triazol-3-yl)benzamide
N-[3-(1H-imidazol-1-yl)propyl]-3-{[(5-methylthiophen-2-yl)methyl]amino}-5-(pyrrolidine-1-sulfonyl)benzamide
5-(2-fluorophenyl)-N-methyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(1-benzothiophene-2-carbonyl)-N-(3-fluorophenyl)piperidin-3-amine
3-[(2R,3R,6R)-5-(dimethyl-1,3-thiazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
6-(azepan-1-yl)-N-(pyridin-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-(furan-2-ylmethyl)-4-(1H-imidazol-1-yl)-N-(pyridin-2-ylmethyl)benzamide
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2,3-dimethoxy-N-{[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-3-yl]methyl}benzamide
2-[1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-yl]ethan-1-ol
1-[(3-fluorophenyl)methyl]-3-(3-methylthiophene-2-carbonyl)piperidine
4-{3-[benzyl(methyl)amino]piperidine-1-carbonyl}-1,2-dihydrophthalazin-1-one
N,6-dimethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-5-carboxamide
(1S,5R)-6-(2,3-difluorobenzoyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
3-(1-tert-butyl-4-phenyl-1H-pyrazol-5-yl)-1-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
5-{2-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(furan-2-yl)-2-oxoacetamide
1-{4-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]piperazin-1-yl}-2,2-dimethylpropan-1-one
N-benzyl{[4-(1H-imidazol-1-yl)phenyl]amino}sulfonamide
6-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pyridine-2-carboxamide
N-ethyl-2-methyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
1-methyl-3-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)-1-(1,2,3,4-tetrahydronaphthalen-1-yl)urea
6-[2-(furan-2-yl)azepane-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
5-[(4-benzylpiperidin-1-yl)methyl]-N-[2-(1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
2-(dimethylamino)-N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}acetamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
{[5-(2-chlorophenyl)furan-2-yl]methyl}({3-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl})amine
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1-cyclobutanecarbonylpiperidine-4-carboxamide
5-(3-fluorophenoxymethyl)-N-(3-hydroxypropyl)-N-methyl-1H-pyrazole-3-carboxamide
1-(4-{[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]amino}-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
4-[2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]benzene-1-sulfonamide
1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazole
[(2S,6S)-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
3-[2-(dimethylamino)ethyl]-8-(2,6-dimethylpyrimidine-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
[(4-methanesulfonylphenyl)methyl](methyl){2-[2-(prop-2-en-1-yl)phenoxy]ethyl}amine
ethyl 1-(thiolan-3-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-methylbenzoyl)piperidine
1-ethyl-4-{5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
3-({2-[2-(2-methylphenyl)pyrimidin-5-yl]-1H-imidazol-1-yl}methyl)-1λ6-thiolane-1,1-dione
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)oxane-4-carboxamide
2-(methylsulfanyl)-5-[(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)methyl]pyrimidine
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(cyclopent-2-en-1-yl)ethan-1-one
1-cyclopropyl-6-oxo-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-N-(propan-2-yl)piperidine-3-carboxamide
3-({[3-(1H-pyrazol-1-yl)phenyl]methyl}amino)pyrazine-2-carbonitrile
N-[3-(4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]-4-fluorobenzene-1-sulfonamide
4-[4-(2,2-dimethylpropyl)piperazin-1-yl]-2-{[4-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
4-[(1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}pyrrolidin-3-yl)methyl]benzoic acid
ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]{[4-methoxy-3-(methoxymethyl)phenyl]methyl}amine
1-ethyl-N,3,5-trimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-4-carboxamide