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N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-cyclopropyl-3-[2-(3-methoxypiperidin-1-yl)-2-oxoethyl]-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
1-[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-[(3-methoxyphenyl)methyl]piperazine
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{5H,6H,7H,8H,9H,10H-cyclohepta[b]indol-2-ylmethyl}-2-(2-ethyl-1H-imidazol-1-yl)acetamide
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-1-(propan-2-yl)piperidine
4-{1-[(4-fluorophenyl)methyl]piperidin-3-yl}-5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidine
N-[(3,5-dimethoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)-5-oxohexanamide
N-[(3-hydroxypyrrolidin-3-yl)methyl]-2-phenoxybenzamide
(3R,4S)-4-cyclopropyl-1-[2-(trifluoromethyl)benzenesulfonyl]pyrrolidin-3-amine
1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
2-{5-oxo-3-[1-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-4-yl}acetic acid
2-methoxy-N-(1-{3-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]phenyl}-1H-pyrazol-4-yl)acetamide
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-fluoro-N-methyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1H-1,3-benzodiazole-2-carboxamide
2-{1-cyclopentyl-4-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]piperazin-2-yl}ethan-1-ol
3-{[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]sulfonyl}-N-methylbenzamide
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]acetamide
1-(2-{[(3R,4R)-1-(benzenesulfonyl)-4-hydroxypyrrolidin-3-yl]amino}ethyl)imidazolidin-2-one
4-[5-(1-methyl-1H-pyrazole-5-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
1-(cyclohex-3-en-1-ylmethyl)-3-(1H-pyrazol-5-yl)piperidine
N-{1-[4-(3-chlorophenyl)-5-[(cyclohexylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}cyclopropanecarboxamide
2-(4-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
4-[2-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]-2-methoxypyridine-3-carbonitrile
3-{imidazo[1,2-a]pyridin-2-yl}-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]propan-1-one
2-(4-{[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}phenoxy)acetic acid
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-3-phenyl-N-(pyrazin-2-ylmethyl)propanamide
methyl (1R,3S,3aR,6aS)-3-[2-(benzyloxy)phenyl]-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
4-(8-hydroxyquinolin-2-yl)-7-(2-oxoimidazolidin-1-yl)-1,2,3,4-tetrahydroquinolin-2-one
1-(2-methoxyphenyl)-2-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
methyl 3-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-1-(2-methoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
2-[(3,5-difluorophenyl)methyl]-8-(1H-imidazol-4-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[1-(3-methoxyphenyl)ethyl]methylamine
4-[3-(2-phenylethyl)-1,2-oxazole-5-carbonyl]-3,4-dihydro-2H-1,4-benzoxazine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]pyrazolo[1,5-a]pyridine-3-carboxamide
8-(2,2-dimethylbutanoyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-{2-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
7-(3-chlorophenyl)-4-(5-propylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2R,3R,6R)-3-(4-fluorophenyl)-5-(piperidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(3-{[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-1H-indazole
4-hydroxy-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-[(phenylsulfanyl)methyl]pyrimidine-5-carboxamide
N-[4-(2-methanesulfonylacetamido)phenyl]-5-methylfuran-3-carboxamide
N-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-{3-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-2-methylpropan-1-one
1-[2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)acetyl]piperidine-4-carboxamide
3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)sulfonyl]-N-(oxolan-2-ylmethyl)benzamide
N-[3-(cyclohexylsulfanyl)propyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
(1S,6R)-9-(5-chloro-3-phenyl-1H-indole-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
4-[5-(2-aminoethyl)-2-methoxyphenyl]phenol
N-ethyl-1-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,3-benzotriazole-5-carboxamide