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N-(2,3-dihydro-1H-inden-2-yl)-N-propyl-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
(3R,4R)-1-(4-methylbenzoyl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
(2E)-N-[(3-methyl-7-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(thiophen-2-yl)prop-2-enamide
2-cyclopentyl-N-{3-[4-({[1-(2-methylpropyl)piperidin-4-yl]methyl}amino)piperidin-1-yl]phenyl}acetamide
3-[(2-methoxyethyl)(methyl)amino]-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-(oxan-4-yl)piperidine-3-carboxamide
3-{[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-5-(propan-2-yl)-1H-pyrazole
1-{6-[2-(hydroxymethyl)phenyl]-1,2,3,4-tetrahydroquinolin-1-yl}ethan-1-one
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-3-(2-methoxyphenyl)propanamide
1-[1-(3-phenylpropyl)piperidin-4-yl]-4-(pyrrolidine-1-carbonyl)piperidine
N-[(4-fluorophenyl)methyl]-3-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}propanamide
5-methyl-1'-(quinoxaline-6-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
(3S,9aR)-3-(cyclohexylmethyl)-8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-ethyl-3-(2-methylpropyl)-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
({3-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)diethylamine
3-{[3-(2,6-dimethylphenoxy)azetidin-1-yl]methyl}pyrrolidine
4-(4-chlorophenoxy)-1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidine
6-(2-fluoro-4-methoxyphenyl)-7-methyl-8-oxo-N-(piperidin-4-ylmethyl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-(oxan-4-yl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2,3,6-trimethylquinoline-4-carboxamide
{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(thiophen-2-yl)ethyl]amine
1-{2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
4-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-1-(2-methoxyphenyl)piperazin-2-one
ethyl 4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
1-[(2-aminopyridin-3-yl)methyl]-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1,4-diazepane-6-carboxylic acid
2-[3-cyclopropyl-5-(1-methyl-5-phenyl-1H-pyrrol-2-yl)-1H-1,2,4-triazol-1-yl]acetic acid
1-[(1-ethylpiperidin-3-yl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane
2-[4-(quinazolin-4-yl)piperazin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
phenyl(1-{[1-(pyrazin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
(3aR,6aR)-2-methyl-N-[2-(quinolin-8-yloxy)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[2-hydroxy-2-(4-hydroxyphenyl)ethyl]-2-(1-propylpiperidin-4-yl)acetamide
N-cyclopentyl-6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridazin-3-amine
4-({[2-amino-6-methyl-5-(prop-2-en-1-yl)pyrimidin-4-yl]amino}methyl)phenol
1-[(2E)-3-phenylprop-2-en-1-yl]-4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperazine
2-(benzyloxy)-1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
2-methyl-2-(naphthalen-1-yloxy)-1-[2-(trifluoromethyl)morpholin-4-yl]propan-1-one
5-[3-cyclopropyl-1-(3,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl]-1H-1,2,4-triazol-3-amine
N'-(2-ethoxyphenyl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]propanediamide
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[(2S)-1-hydroxypropan-2-yl]acetamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(1R)-2-hydroxy-1-phenylethyl]propanamide
(4aS,8aS)-2-[(1-methyl-1H-indol-5-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
2-(1-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)pyridine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
1-{[3-(methylsulfanyl)phenyl]methyl}-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-(1-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-1-oxopentan-2-yl)acetamide
4-{[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]methyl}-N,N-dimethyloxan-4-amine
N-[(4-hydroxyphenyl)methyl]-N-(pyridin-3-ylmethyl)oxane-2-carboxamide
1-[2-methoxy-4-({[(3-methylphenyl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol