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(2S,4R)-4-amino-N-methyl-1-{2-methyl-3-[(pyridin-3-ylmethyl)amino]benzoyl}pyrrolidine-2-carboxamide
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-(2-methoxyethyl)-N-(propan-2-yl)propanamide
1-({3-[2-(thiophen-2-yl)azetidine-1-carbonyl]phenyl}methyl)-1H-pyrazole
4-[(1-ethyl-1H-imidazol-2-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(quinolin-3-yl)benzamide
1-[(diethylcarbamoyl)methyl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(2-methylphenyl)-4-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)piperazine
2-[2-(4,4-difluoropiperidin-1-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
2-(3-methoxypropyl)-8-(pyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
(2S)-4-methanesulfonyl-2-{[5-(propan-2-yl)-1,2-oxazol-3-yl]formamido}butanoic acid
N-(1-hydroxy-2-methylpropan-2-yl)-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-methyl-3-propyl-N-(quinolin-2-ylmethyl)-1H-pyrazole-5-carboxamide
4-{[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-methyl-1H-pyrazole
3-ethyl-4-methyl-N-(4-phenylbutyl)-1H-pyrazole-5-carboxamide
1-[4-({3-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
N-(2,1,3-benzoxadiazol-4-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-amine
3-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
1-[(1,3-dimethyl-1H-pyrazol-5-yl)sulfonyl]-3-methyl-3-phenylpiperidine
4-[(4-fluorophenyl)methyl]-1-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
3-(3-cyclohexyl-1H-1,2,4-triazol-5-yl)-1-[(3-methylpyridin-4-yl)methyl]urea
(1S,3R)-3-amino-N-methyl-N-(quinoxalin-2-ylmethyl)cyclopentane-1-carboxamide
1-[4-(4-benzylpiperazin-1-yl)piperidin-1-yl]-2-(morpholin-2-yl)ethan-1-one
N-[(2-ethoxy-3-methoxyphenyl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
7-fluoro-N-(1,2-oxazol-3-ylmethyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-{[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}benzoic acid
N-[(1R,3R)-3-aminocyclopentyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
9-oxo-N-(4-phenylphenyl)-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(propan-2-yloxy)propan-1-one
3-{2-[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}-5-(oxolan-2-yl)-1,2,4-oxadiazole
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[(2-hydroxyethyl)(methyl)amino]methyl}piperidin-2-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}acetamide
1-{[3-(2,3-dihydro-1H-isoindole-2-carbonyl)-1H-pyrazol-5-yl]methyl}-1H-1,3-benzodiazole
1-(5-ethyl-1,2-oxazole-4-carbonyl)-3-(3-methylphenoxymethyl)piperidine
N-(3-{4-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}propyl)oxolane-2-carboxamide
(1-{[1-(1-methyl-1H-imidazole-2-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanamine
N-[(2-chlorophenyl)methyl]-3-[1-(4,4,4-trifluorobutanoyl)piperidin-3-yl]propanamide
2-(methylamino)-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
N-[1-(7-{[3-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-2-carboxamide
N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
4-(1-benzothiophene-5-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
3-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}-N-(propan-2-yl)propanamide
6-{4-[(8-chloroquinolin-2-yl)methyl]piperazin-1-yl}pyrimidine-2,4-diamine
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-N-methyl-N-(1-methylpiperidin-4-yl)-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-(6-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-{1-[(5-phenylthiophen-2-yl)methyl]piperidin-3-yl}propanamide
N-[(2-fluorophenyl)methyl]-3-(1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)propanamide
N-(2-{1-[(4-methylphenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}ethyl)furan-2-carboxamide
(1R,5R)-6-[2-(ethylamino)pyrimidine-5-carbonyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-benzyl-2-(ethanesulfonyl)-N-methyl-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide