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3-[(methylamino)methyl]-4-(2-phenoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-ethyl-2-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-6-(piperidin-3-yl)pyrimidin-4-amine
N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-4-(pyridin-3-yl)pyrimidin-2-amine
2-(1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethan-1-ol
[1-(2,3-difluoro-4-methoxybenzoyl)-3-propylpiperidin-3-yl]methanol
5-acetyl-N-(furan-2-ylmethyl)-N-(prop-2-en-1-yl)thiophene-2-carboxamide
8-(6-chloropyridazin-3-yl)-2,8-diazaspiro[4.5]decan-3-one
1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-4-phenylbutane-1,4-dione
4-[5-(methoxymethyl)thiophene-2-carbonyl]-2-[(4-methoxyphenyl)methyl]morpholine
5-methyl-N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-[(3-methoxyphenyl)methyl]-N-methyl-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
4-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1,2,4-oxadiazol-3-yl}-1H-indole
1-{4-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-4-oxobutyl}pyrrolidin-2-one
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-2-(2-oxopyrrolidin-1-yl)acetamide
N-[(2-aminopyridin-3-yl)methyl]-2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
2-[1-(furan-2-ylmethyl)-4-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
4-[1-(2-phenylethyl)-5-(pyridine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
2-(1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-2-yl)-6-methyl-1H-1,3-benzodiazole
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-(ethylamino)pyrimidine-5-carboxamide
(3S,4S)-1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
5-[(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)methyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-5-[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazole
(3S,4S)-4-cyclopropyl-1-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)pyrrolidine-3-carboxylic acid
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)pyrimidin-4-amine
3,4,7-trimethyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-1H-indole-2-carboxamide
5-(4-formylpiperazin-1-yl)-1-methyl-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-(3,6-dimethyl-1-benzofuran-2-carbonyl)-N-methyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
N,N-dimethyl-2-{[(3-phenyl-1,2,4-oxadiazol-5-yl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
3-chloro-N-[4-methoxy-2-(2-methylpropanamido)phenyl]pyridine-4-carboxamide
2-(benzyloxy)-1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}ethan-1-one
4-amino-N-[3-(2,6-dimethylphenoxy)propyl]-N-methylpyridine-2-carboxamide
N'-(3-ethylphenyl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)butanediamide
ethyl 4-(2-methoxyethyl)-1-[(2,4,5-trimethoxyphenyl)methyl]piperidine-4-carboxylate
4-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
N-cyclohexyl-1-cyclopropyl-4-oxo-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
1-[(2S)-2-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]pyrrolidin-1-yl]ethan-1-one
N,5-dimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
2-(dimethyl-1,2-oxazole-4-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-({1-[(4-methylphenyl)methyl]piperidin-3-yl}methyl)-2-(1H-1,2,4-triazol-1-yl)acetamide
2-[(3,5-difluorophenyl)methyl]-8-(2-methoxybutanoyl)-2,8-diazaspiro[4.5]decan-3-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
3-{2-[2-(dimethylamino)-2-(2-methylphenyl)acetamido]acetamido}propanoic acid
(3R,4S)-1-{4-[(diethylamino)methyl]-5-ethylfuran-2-carbonyl}-3,4-dimethylpiperidin-4-ol
(3-{[ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-2,4,6-trimethylphenyl)methanol
2-[(1-ethylpyrrolidin-3-yl)methyl]-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
2-(3-chlorophenyl)-N-{2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}acetamide
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one