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2-fluoro-N-[(3-methyl-7-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
11-{[2-(methylsulfanyl)ethyl]amino}-4-{[3-(trifluoromethyl)phenyl]methyl}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[(1-phenylmethanesulfonylpiperidin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
2-[2-(1H-imidazol-4-yl)ethyl]-8-(pyrimidin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(4-methoxyphenyl)methyl]piperidine
3-(1-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methoxyphenyl)urea
2-{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethoxy}acetamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-4-(trifluoromethyl)benzamide
6-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidin-4-amine
4-fluoro-3-[1-(2-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]benzene-1-sulfonamide
7-(3-chlorophenyl)-4-(pyrrolidine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(2-fluorophenyl)-2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidine-6-carboxamide
3-[1-(3-hydroxypyridine-4-carbonyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
2-[2-(3-fluorophenyl)azepane-1-carbonyl]-3,5-dimethyl-1H-indole
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-oxo-4H-chromene-2-carboxamide
N-[(2-methoxyquinolin-3-yl)methyl]-1-(pyrimidin-2-yl)piperidin-3-amine
(2R,3R)-3-amino-1'-(1H-indole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-benzyl-4-chloro-N-(1,1-dioxo-1λ6-thiolan-3-yl)-1-methyl-1H-pyrazole-3-carboxamide
ethyl 1-[2-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamido]cyclobutane-1-carboxylate
4-(6-aminopyridine-3-carbonyl)-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(2-oxo-2-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}ethyl)-1,2-dihydroisoquinolin-1-one
(2S)-2-({[bis(prop-2-en-1-yl)carbamoyl]methyl}amino)-3-methylbutanamide
1-[2-(2,4-difluorophenyl)acetyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
4-hydroxy-N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2-(phenoxymethyl)pyrimidine-5-carboxamide
(3R,4R)-4-(azepan-1-yl)-1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-ol
2-(1-{[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}-3-oxopiperazin-2-yl)-N-methylacetamide
2-(2-hydroxyethyl)-8-(quinoline-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
5-(1-methyl-1H-imidazol-2-yl)-1-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-4-phenyl-1H-imidazole
1-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
[4-({1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
3-{ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]amino}-1λ6-thiolane-1,1-dione
N-[3-(3,5-dimethylphenoxy)propyl]-N-methyl-2-(pyridin-3-yloxy)acetamide
1-(3-{3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4H-1,2,4-triazol-4-yl}phenyl)ethan-1-one
3-({[2-(dimethylamino)ethyl][(2-methylphenyl)methyl]amino}methyl)-7-fluoro-1,2-dihydroquinolin-2-one
3-(4-chlorophenyl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-phenylpropanamide
6-chloro-2-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonan-7-yl}methyl)-1,4-dihydroquinolin-4-one
(3S,4S)-N-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-methoxy-1-(propan-2-yl)pyrrolidin-3-amine
2-(4-{[4-(4-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]methyl}phenyl)acetic acid
5-cyclobutanecarbonyl-1'-(3,3,3-trifluoro-2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[2-({6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl}formamido)ethyl]piperidine-3-carboxamide
2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-N,N-dimethylpyridine-3-carboxamide
2-phenyl-5-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}pyrimidine
2-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]acetic acid
7-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-{[4-(trifluoromethoxy)phenyl]methyl}imidazo[1,2-a]pyridine-6-carboxamide
2-[1-(2-methyl-1,3-benzothiazol-6-yl)-5-[(methylamino)methyl]-1H-1,2,4-triazol-3-yl]acetamide
[(dimethyl-1,2-oxazol-4-yl)methyl]({2-[(3-fluorophenyl)methoxy]-3-methoxyphenyl}methyl)methylamine
N-[5-(4-methylphenyl)-1,3,4-thiadiazol-2-yl]-4-(3-methylpyridin-4-yl)piperazine-1-carboxamide
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}oxolane-2-carboxamide