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[(2,4-dimethoxypyrimidin-5-yl)methyl](methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
(1S,5R)-3-[6-amino-2-(methylsulfanyl)pyrimidin-4-yl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-[4-(1H-indol-2-ylmethyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[3-(2-phenylethyl)piperidin-1-yl]ethan-1-one
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(4H-1,2,4-triazol-4-yl)piperidine
5-cyclopropanecarbonyl-1'-(1-ethylpiperidine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(4aS,7aR)-1-(2-aminoacetyl)-4-benzyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(diethylamino)ethyl]-1-[2-(2-methoxyethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-4-carboxamide
dimethyl[1-(4-{6-methylthieno[2,3-d]pyrimidin-4-yl}phenyl)ethyl]amine
3-{1-[(2-propyl-1,3-thiazol-4-yl)methyl]-1H-1,2,3-triazol-4-yl}benzonitrile
2-[4-(3-fluorophenyl)-1H-pyrazol-1-yl]-N-{1-[(5-methylfuran-2-yl)methyl]-1H-pyrazol-5-yl}acetamide
4-benzyl-3-ethyl-1-[(3-methylpyridin-2-yl)methyl]-1,4-diazepan-5-one
4-{pyridin-3-yl[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}morpholine
2-[(2-phenylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
(1R,3S)-7-(2-methyl-4-phenylpyrimidine-5-carbonyl)-7-azaspiro[3.5]nonane-1,3-diol
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(4-methyl-1H-pyrrole-2-carbonyl)pyrrolidin-3-yl]methanol
3,5-dimethoxy-2-[(2-methyl-3-oxopiperazin-1-yl)methyl]benzoic acid
2-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-5,6-dimethylpyridine-3-carbonitrile
2-(2-chloro-6-fluorophenyl)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
2-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-5-(propan-2-yl)furan-3-carboxamide
4-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]thiomorpholine
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(2-hydroxyethyl)piperazin-1-yl]ethan-1-one
3-(3,4-difluorophenyl)-N-methyl-N-(pyrazin-2-ylmethyl)propanamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-2-phenyl-1,3-thiazole
4-[3-fluoro-5-(trifluoromethyl)phenyl]-6-(morpholin-4-yl)pyrimidin-2-amine
(1S,5R)-6-benzyl-3-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(1,3-thiazol-2-ylmethyl)piperidine
6-methyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-2H-1,3-benzodioxol-5-amine
2-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}pyridine-3-carboxylic acid
2-(dimethylamino)-4-methyl-N-[(4-sulfamoylphenyl)methyl]pyrimidine-5-carboxamide
1-(2-chloro-5-fluorophenyl)-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-methylurea
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(propylsulfanyl)acetyl]pyrrolidine-3-carboxylic acid
3-(1-methyl-1H-pyrazol-4-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-methyl-1-[2-(pyridin-2-yl)ethyl]urea
3-{1-[3-(3-methoxyphenyl)-1H-pyrazol-5-yl]-N-methylformamido}propanamide
2-(2-aminoethyl)-5,6-dimethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}thieno[2,3-d]pyrimidin-4-amine
2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]morpholine-4-carboxamide
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-methoxypyridine
2-[3-benzyl-1-(2-chlorophenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-methylacetamide
N-(1-cycloheptylpiperidin-3-yl)cyclobutanecarboxamide
butyl (4aS,7aR)-6,6-dioxo-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
3-[1-(carbamoylmethyl)-1H-imidazol-2-yl]-N-(cyclohexylmethyl)piperidine-1-carboxamide
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(methoxymethyl)-1H-pyrazole-4-carbonyl)-4-methylpiperazine
7-methyl-2-[(2-methylpyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-methyl-1-[3-(methylsulfamoyl)phenyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)urea
N-[1-(3-methylphenyl)piperidin-4-yl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
4-{1-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]ethyl}morpholine
6-{3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one