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1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
[(3R,4R)-1-(4-methoxy-2-methylbenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-(1H-imidazol-1-ylmethyl)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-ol
2-(4-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]ethan-1-one
3-{1-[3-(1H-pyrazol-1-yl)benzoyl]azetidin-3-yl}pyridine
5-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(3S,4R)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
7-(cyclohexylmethyl)-2-(3-methylfuran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-[(4-butylpiperazin-1-yl)methyl]-7-chloro-1,2-dihydroquinolin-2-one
dimethyl({5-[2-(4-methylpentyl)morpholine-4-carbonyl]furan-2-yl}methyl)amine
5-(dimethylamino)-2-({6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,3-dihydropyridazin-3-one
N-(cyclopropylmethyl)-2-methyl-N-(propan-2-yl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(2R,3R,6R)-3-(4-fluorophenyl)-5-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
propan-2-yl 4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
3-{[4-(3-chloro-4-fluorophenyl)-1H-1,2,3-triazol-1-yl]methyl}-N,N-dimethylbenzamide
1-{5-[3-(1H-pyrazol-3-yl)phenyl]thiophen-2-yl}propan-1-one
1-benzyl-8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(2,5-di-tert-butylphenyl)-1-[3-(3-oxopiperazin-1-yl)propyl]urea
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-{imidazo[1,2-b]pyridazin-6-yl}piperazine
(1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-4-[(3-methoxyphenyl)methyl]piperidin-4-yl)methanol
N-[(2-methoxyphenyl)methyl]-2-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)acetamide
N-benzyl-N-ethyl-3-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]propanamide
N-{2-[1-(1,2-dihydroacenaphthylen-5-yl)-1H-imidazol-4-yl]ethyl}acetamide
methyl 1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperidine-2-carboxylate
3-methoxy-2,2-dimethyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propanamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(cyclohex-3-ene-1-carbonyl)-7-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
benzyl({[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})methylamine
N-methyl-2-{2-methylimidazo[1,2-a]pyridin-3-yl}-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
6-(benzyloxy)-4-(furan-3-ylmethyl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
4-(4-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperazine-1-carbonyl)morpholine
N-cyclopentyl-3-ethyl-1-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1H-pyrazole-5-carboxamide
N-[(1-methylpiperidin-4-yl)methyl]-4-oxo-N-(2-phenylethyl)-3,4-dihydrophthalazine-1-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-dimethylacetamide
4-benzyl-3-{2-oxo-2-[4-(quinazolin-4-yl)piperazin-1-yl]ethyl}piperazin-2-one
{[2-chloro-5-ethoxy-4-(propan-2-yloxy)phenyl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
2-phenyl-1-(1-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)ethan-1-ol
N-[3-(3-fluorophenyl)phenyl]-1-(1-propylpiperidin-4-yl)piperidine-4-carboxamide
[5-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)furan-2-yl]methanol
(1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-4-yl)methanol
1-[3-(4-acetyl-6-hydroxy-1,4-diazepane-1-carbonyl)phenyl]pyrrolidin-2-one
2-(2-chloro-6-methoxy-4-{6-oxa-9-azaspiro[4.5]decan-9-ylmethyl}phenoxy)acetamide
3,6-dimethyl-N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-1-benzofuran-2-carboxamide
N-[2-(4-hydroxy-3-methoxyphenyl)ethyl]-5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(2-hydroxyethyl)pyrrolidin-3-yl]-5-fluoro-2-methoxybenzamide
6-[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]pyridine-2-carbonitrile
1-[1-(4-chloro-2-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
N-[2-(propylsulfanyl)ethyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
5-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]methyl}-1-phenyl-1H-1,2,3,4-tetrazole