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2-methoxy-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}-2-phenylethan-1-one
[(4-chlorophenyl)methyl]({[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl})amine
4-{4-[(4-fluorophenyl)methyl]piperazin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[3-({[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]carbamoyl}amino)phenyl]acetamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(pyridin-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
{3-[(3-chlorophenyl)methyl]-1-(pyridin-3-ylmethyl)piperidin-3-yl}methanol
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(2-phenylethyl)benzamide
2-(cyclopropylamino)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]acetamide
5,6-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidin-4-amine
2-methoxy-5-({4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}methyl)phenol
3-(1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
N,N-bis(1,3-oxazol-4-ylmethyl)-5,6,7,8-tetrahydroquinoline-3-carboxamide
2-{[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](methyl)amino}-N,N-dimethylpropanamide
4-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
5-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-{1-[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl]pyrrolidin-3-yl}-N-ethylacetamide
methyl({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}){[2-(trifluoromethyl)phenyl]methyl}amine
1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-(5,5-dimethyl-2,4-dioxoimidazolidin-1-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}acetamide
(2-{7-[(2,3-dimethoxyphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)urea
N-{1-[1-(2-hydroxyacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
4-{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}piperazin-2-one
4-(1H-1,3-benzodiazol-2-ylmethyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
2-(4-methyl-1,4-diazepan-1-yl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethan-1-one
8-(2-hydroxy-3-methylbenzoyl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(pyridin-2-yl)ethyl]amine
N-{3-methyl-1-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]butyl}thiophene-2-carboxamide
N-ethyl-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
4-(1-benzothiophen-2-ylmethyl)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-{2H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5-{5-[(2,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
4-[3-(1H-pyrazol-5-yl)phenyl]-4H-1,2,4-triazole
5-(benzenesulfonyl)-3-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5-cyclopropanecarbonyl-1'-(pyridine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{1-cyclopentyl-4-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
N4-methyl-6-(morpholin-4-yl)-N4-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrimidine-2,4-diamine
N-(2-hydroxyethyl)-2-methoxy-N-(1,3-thiazol-2-ylmethyl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-chloro-4-({3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)pyridine
4-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-6-methylquinoline
5-ethyl-3-{2-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,2,4-oxadiazole
5-[1-(piperidin-1-yl)ethyl]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}furan-2-carboxamide
3-{2-[4-(3,4-dichlorophenyl)piperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
N-(2-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}quinolin-5-yl)acetamide
5-{[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]sulfonyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
(1S,3R)-3-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}cyclohexan-1-amine
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
5-{2-[2-(dimethylamino)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(4-chlorophenyl)-N-{[1-(pyridin-4-yl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
2-ethoxy-6-{[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]methyl}phenol