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N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}cyclohex-3-ene-1-carboxamide
4-(2-phenylbenzoyl)-1,4-oxazepan-6-ol
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(2R,6S)-2,6-dimethyl-4-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}morpholine
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[2-methyl-4-oxo-1-(oxolan-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
(2S,4R)-1-benzyl-N-ethyl-4-[2-(3-methyl-1,2-oxazol-5-yl)acetamido]pyrrolidine-2-carboxamide
3-{1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidin-3-yl}propanamide
ethyl 1-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)piperidine-3-carboxylate
2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
4-benzyl-1-(2-ethoxyacetyl)-3-ethyl-1,4-diazepan-5-one
5-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridin-3-amine
5-{2-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}-2-methylpyridine
N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}-1H-indole-3-carboxamide
4-{5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]furan-2-yl}-2-methylbut-3-yn-2-ol
4-{1-[3-(1H-pyrazol-4-yl)propyl]piperidin-4-yl}thiomorpholine
3-methyl-7-({1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}methyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-{3-[(dimethylamino)methyl]-1,2,4-oxadiazol-5-yl}-2-methyl-N-(pyridin-3-ylmethyl)aniline
N-methyl-6-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
N-(2,6-dimethylphenyl)-3-[(3,4-dimethylphenyl)amino]piperidine-1-carboxamide
(3R,5S)-5-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrrolidin-3-ol
2-{4-[2-(4-chlorophenoxy)ethyl]phenyl}-N-methylacetamide
8-(6-chloropyridazin-3-yl)-2-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(2-methanesulfonylethyl)-4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazine
(3R,5S)-5-(3-fluorophenoxymethyl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]-1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(3S,4S)-4-methyl-1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidine-3,4-diol
4-{4-[3-(2-hydroxyethyl)-4-methylpiperazine-1-carbonyl]phenyl}-2-methylbutan-2-ol
(1S,5R)-6-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
1-cyclopentanecarbonyl-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylpiperidine-4-carboxamide
2-(ethoxymethyl)-N-{1-oxaspiro[4.4]nonan-3-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methylbenzamide
methyl 5-(cyclobutylamino)-3-(4-methoxybenzamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
8-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-1,3-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-methyl-7-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(2S,4R)-4-amino-1-[2,4-bis(trifluoromethyl)benzoyl]-N-methylpyrrolidine-2-carboxamide
1-[2-(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
ethyl 1-[5-(methoxymethyl)thiophene-2-carbonyl]-3-(2-phenylethyl)piperidine-3-carboxylate
3-(phenoxymethyl)-5-[3-(4H-1,2,4-triazol-4-yl)phenoxymethyl]-1,2,4-oxadiazole
N-cyclopropyl-5-methyl-1-propyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
3-ethyl-8-[(6-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-[(3-methyl-1H-pyrazol-4-yl)methyl]-4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
(4aS,8aS)-2-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-decahydroisoquinolin-4a-ol
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(propan-2-yl)piperidine-3-carboxamide
9-[2-(1H-imidazol-1-yl)acetyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(morpholine-4-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
2-chloro-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzene-1-sulfonamide
1-{3-[benzyl(methyl)amino]piperidin-1-yl}but-2-yn-1-one
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-(thian-4-yl)piperazine
(4aS,8aR)-6-(2-hydroxyacetyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one