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N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]cyclohexanecarboxamide
1-{3-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
2-{4-[(2-ethylphenyl)methyl]-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl}acetic acid
(2R,3R,6R)-5-(2H-1,3-benzodioxole-5-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(3-methoxypropyl)-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N'-(3,5-difluorophenyl)-N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}ethanediamide
(3R,4S)-4-cyclopropyl-1-[8-(trifluoromethyl)quinolin-4-yl]pyrrolidin-3-amine
3-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-ylmethyl]-N-(2-methoxy-6-methylphenyl)benzamide
N-[(1R,3R)-3-aminocyclopentyl]-2-hydroxy-3-methylbenzamide
N-[1-(1H-1,3-benzodiazol-2-yl)-3-(methylsulfanyl)propyl]-5-propyl-1,2-oxazole-3-carboxamide
[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl](methyl){[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
1-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-methoxyethan-1-one
N-{2-[1-(furan-2-ylmethyl)piperidin-3-yl]ethyl}-1,3-thiazole-5-carboxamide
3-{5-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]-4-phenyl-1H-imidazol-1-yl}propan-1-ol
1-[(3-methoxyphenyl)methyl]-4-(4-methyl-1H-pyrrole-2-carbonyl)piperazin-2-one
4-methyl-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-1H-imidazole-5-carboxamide
1-(4-fluorophenyl)-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}piperazine
5-cyclopropanecarbonyl-1'-(5-methyl-1,2-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-benzyl-3-ethyl-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1,4-diazepan-5-one
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(quinoline-8-sulfonamido)acetic acid
2-phenyl-1-{1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-4-yl}ethan-1-ol
1-[2-(4-methoxyphenyl)ethyl]-5-{2-[(2-phenoxyethyl)amino]ethyl}pyrrolidin-2-one
2-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
(1R,5R)-6-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
3-(2-chlorophenyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3-phenylpropanamide
N-(4-chloro-2-methylphenyl)-3-[3-(trifluoromethyl)benzoyl]piperidine-1-carboxamide
5-{1-[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]ethyl}-2-methylpyridine
3-(3-fluorophenyl)-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-4-carboxamide
2-methoxy-5-[2-(2-phenyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]benzamide
9-[(2S)-2-amino-2-phenylacetyl]-2-[3-(dimethylamino)propyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
1-(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)ethan-1-ol
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)cyclopropanecarboxamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-methanesulfonyl-N-[1-(4-methylphenyl)-5-oxopyrrolidin-3-yl]acetamide
5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[(3-methyloxetan-3-yl)methyl]-1,2-oxazole-3-carboxamide
2-oxo-N-[3-(1H-pyrazol-5-yl)phenyl]-1,3-dioxa-8-azaspiro[4.5]decane-8-carboxamide
4-phenyl-N-({1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidin-3-yl}methyl)benzamide
6-{[5-(4-fluorophenyl)-1,2,4-triazin-3-yl]amino}-2-methylheptan-2-ol
N'-(2-ethoxyphenyl)-N-methyl-N-(quinolin-4-ylmethyl)propanediamide
N-{1-[1-(5-acetylthiophene-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-3-methoxy-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
2-methoxy-3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
1-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]naphthalen-2-ol
3-[(4aS,7aR)-4-(2-hydroxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
2-({1-[(2-methoxyethyl)(methyl)amino]hex-5-en-2-yl}oxy)-N-methylpyridine-4-carboxamide
2-(5-fluoro-2-methylphenyl)-N-[1-(pyridin-2-yl)propyl]acetamide
1-{3-[9-methoxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]phenyl}pyrrolidin-2-one
1-(cyclohex-3-ene-1-carbonyl)-4-(3-methylpyridin-2-yl)piperazine