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2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
4-(4-methylpiperazin-1-yl)-6-[3-(1H-pyrazol-5-yl)phenyl]quinazoline
N-(5-fluoro-2-methylphenyl)-2-{[3-(1H-imidazol-2-yl)phenyl]formamido}acetamide
ethyl 1-[(3-{[1-(pyridine-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]piperidine-2-carboxylate
5-(3-chloro-4-ethoxyphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
(2R,3R)-1'-[6-(dimethylamino)pyrimidin-4-yl]-3-[ethyl(methyl)amino]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
methyl[(6-methylpyridin-2-yl)methyl]{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
1-(2H-1,3-benzodioxole-5-carbonyl)-4-(2-methylquinolin-6-yl)piperidin-4-ol
1-[3-(2-methylphenoxymethyl)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
3-(2-hydroxyethyl)-4-(1-methyl-1H-indazole-3-carbonyl)piperazin-2-one
N-(pyridin-3-yl)-2-[2-(1H-pyrrol-1-yl)propanoyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
(2-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}ethyl)urea
(2S,4R)-1-[(2-methoxynaphthalen-1-yl)methyl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
2-(3-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}phenoxy)acetamide
N-[2-(ethanesulfonyl)ethyl]-3-phenyl-1H-pyrazole-4-carboxamide
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
8-[2-(2,4-difluorophenyl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-N-[(1-methylpiperidin-2-yl)methyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
4-(3,4-difluorophenyl)-1-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1H-1,2,3-triazole
1-[2-(4-methoxyphenyl)ethyl]-N-[(3-methylpyridin-4-yl)methyl]-6-oxopiperidine-3-carboxamide
N-(2-methoxyethyl)-N-(oxolan-2-ylmethyl)-1H-pyrazole-4-carboxamide
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}acetamide
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
N-[4-(2-oxo-2-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}ethyl)phenyl]cyclopropanecarboxamide
5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazole
N-(2-{7-[(3-ethoxy-2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
4-{3-[4-(2-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
(4aS,7aR)-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[1-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperidin-3-yl]pyrimidin-4-ol
1-[2-(piperidin-1-yl)ethyl]-N-[1-(pyrazin-2-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
5-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-4-methylpyrimidine
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
5-[1-(4-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(2R)-1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
9-cyclohexanecarbonyl-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-({1-[4-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazol-1-yl]propan-2-yl}oxy)pyridine
2,3,5-trimethyl-6-[1-(pyridin-3-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]pyrazine
4-(4-chlorophenyl)-3-(oxan-4-yl)-4H-1,2,4-triazole
8-[2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
(1R,2S)-2-{[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}cyclopentane-1-carboxamide
1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(2-hydroxyphenyl)ethan-1-one
1-methyl-4-({5-[(2E)-pent-2-en-1-yl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(pyridin-2-yl)ethyl]amine
2-methyl-6-{4-[3-(trifluoromethyl)phenoxy]piperidine-1-carbonyl}pyridine
N-cyclopropyl-1-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
2-{2-[(1-benzylpyrrolidin-3-yl)amino]ethyl}-1,2-dihydrophthalazin-1-one
1-{1-methyl-5-[(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)methyl]-1H-pyrrol-3-yl}ethan-1-one
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]benzamide