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2-ethyl-8-[3-(4-methyl-1,4-diazepan-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
(2E)-3-(3,4-dimethoxyphenyl)-N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)prop-2-enamide
(1S,5R)-3-benzyl-6-(4-methylpiperazine-1-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
7,7-dimethyl-2-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-[(3-chloropyridin-4-yl)methyl]-2-(pyridin-3-yl)morpholine
N-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(5-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
2-[(4aS,7aR)-4-(2-methoxyacetyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N-(1-methyl-1H-pyrazol-3-yl)acetamide
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine
2-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]pyridine-3-carbonitrile
3-(2-phenylethyl)-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
2-methyl-3-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)quinoxaline
N-methyl-N-[(1-methylpiperidin-3-yl)methyl]-2-(thiophene-2-sulfonamido)acetamide
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-3-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}benzamide
2-{5-[6-amino-5-cyano-4-(5-ethylfuran-2-yl)pyridin-2-yl]thiophen-3-yl}acetic acid
N-cyclopropyl-4-methoxy-2-({1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)benzamide
1-(1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1,4-diazepan-5-one
dimethyl(3-{2-[1-(quinoxalin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(hydroxymethyl)piperidin-3-ol
6-[(2S)-1-hydroxy-4-methylpentan-2-yl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-{[4-(dimethylamino)piperidin-1-yl]methyl}-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
3-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-N-cyclohexylpropanamide
1-(4-{[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
4-{5-[4-(morpholine-4-carbonyl)piperazine-1-carbonyl]-1H-pyrazol-3-yl}phenol
2-({4-[3-(trifluoromethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetic acid
2-(1-benzylpiperidin-3-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(2-{1-[2-(2-hydroxyethyl)phenyl]-1H-imidazol-2-yl}quinolin-6-yl)acetamide
4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}-1-(3-methylpiperidine-3-carbonyl)piperidine
1-(cyclopropylmethyl)-N-ethyl-5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[4-(2-methoxybenzoyl)piperazin-1-yl]-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-methyl-N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
9-(2-methoxyethyl)-1-methyl-10-oxo-N-(propan-2-yl)-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
8-hexanoyl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[2-(methylsulfanyl)benzoyl]piperidine
({4-[1-(2-cyclopropylpyrimidine-5-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
1-(1-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)-2-(4-methoxyphenoxy)ethan-1-one
6-(2,5-dimethylfuran-3-yl)-7-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-(2-benzamido-5-ethylthiophene-3-carbonyl)piperazine-2-carboxylic acid
(4-{[2-(benzyloxy)phenyl]methyl}morpholin-3-yl)methanol
1-[2-(1-methyl-1H-pyrazol-5-yl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)cyclopent-1-ene-1-carboxamide
2-ethyl-8-phenylmethanesulfonyl-2,8-diazaspiro[5.5]undecan-3-one
1-(2,5-dihydro-1H-pyrrol-1-yl)-2-(4-{[4-(pyridin-2-yl)phenyl]methyl}morpholin-3-yl)ethan-1-one
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-(4-fluorophenyl)-1-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)piperidin-3-amine
(3R,4R)-1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol