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N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}cyclobutanecarboxamide
(3S,4S)-1-[6-(propan-2-yl)pyrimidin-4-yl]-4-(propan-2-yloxy)pyrrolidin-3-ol
N-(2,1,3-benzothiadiazol-4-yl)-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
ethyl 4-[10-(methoxycarbonyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-3-yl]piperidine-1-carboxylate
2-(4-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-N,N-dimethylacetamide
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine
1-cyclopentyl-3-(2-methylphenyl)-3-{2-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
N-[(3S,4R)-1-(azepane-1-sulfonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
N-[2-(2-chloro-4-methylphenoxy)ethyl]-N-methyl-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
6-{[5-(5-ethylpyridin-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-2-methylpyrimidin-4-ol
3-{1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl N-{2-[3-(4-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}carbamate
3-{5-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]-4-phenyl-1H-imidazol-1-yl}butanoic acid
3-methyl-6-{2-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-imidazol-1-yl}-2,3-dihydro-1,3-benzoxazol-2-one
3-{[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyridin-2-amine
(3S,4R)-1-(4-fluorobenzoyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N-[(2S)-1-methoxypropan-2-yl]-4-methyl-7-(methylsulfanyl)quinolin-2-amine
4-(4-fluorophenoxy)-1-[(2S)-piperidine-2-carbonyl]piperidine-4-carboxylic acid
3-(4-methoxyphenyl)-N-[(5-methylpyrazin-2-yl)methyl]-3-phenylpropanamide
7-(cyclopropylmethyl)-2-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
2-({4-[(3-methoxyphenyl)methyl]piperazin-1-yl}methyl)-6-methylquinolin-4-ol
4-[(4-fluorophenyl)methyl]-N-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-1,4-diazepane-1-carboxamide
methyl (2S)-2-{[2-(4-fluorophenoxymethyl)-1,3-oxazol-4-yl]formamido}-2-phenylacetate
3-(4-fluorophenyl)-N-[1-(2-methoxyphenoxy)propan-2-yl]-1H-pyrazole-5-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-3-(4-methylphenyl)-1H-pyrazole-5-carboxamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylcyclobutanamine
1-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-3-propyl-1H-pyrazole-5-carboxamide
1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-4-(1-methylpiperidin-4-yl)piperazine
N-[(5-methylfuran-2-yl)methyl]-3-{1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-3-yl}propanamide
(2Z)-2-fluoro-1-[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]-3-phenylprop-2-en-1-one
N-{[2-(4-acetylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-5-methylthiophene-2-carboxamide
1-{2-[(6,8-dimethoxy-4-methylquinolin-2-yl)amino]ethyl}imidazolidin-2-one
2-ethoxy-4-{[methyl({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amino]methyl}phenol
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(1H-pyrrole-2-carbonyl)piperazine
1-(2,6-difluoro-4-methoxybenzoyl)-3-(2-methoxyphenoxy)azetidine
2-(ethylamino)-N-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
N-ethyl-2-[4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)morpholin-3-yl]acetamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(pyrazin-2-yl)propanamide
5-cyclopropanecarbonyl-1'-(3,5-difluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
dimethyl[3-(2-{1-[2-(methylsulfanyl)benzoyl]piperidin-4-yl}-1H-imidazol-1-yl)propyl]amine
1-methyl-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
4-[1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]-3,5-dimethyl-1,2-oxazole
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{2-[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}acetamide
3-{1-[2-(methylamino)pyrimidin-5-yl]-N-(2-phenylethyl)formamido}propanamide
4-[4-(4-fluorophenyl)butanoyl]-1-phenylpiperazin-2-one
(1S,5R)-6-(cyclobutylmethyl)-3-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(4-{[2-(4-fluorophenyl)phenyl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[4-(8-methoxyquinolin-2-yl)-1H-pyrazol-1-yl]acetamide
{1-[2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)ethyl]piperidin-3-yl}methanol