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{[3-(4-fluorophenyl)oxolan-3-yl]methyl}({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
3-({[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
(4aR,8aR)-7-(4,6-dimethylpyrimidin-2-yl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
ethyl 1-[1-(1,3-dioxo-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindol-4-yl)piperidine-4-carbonyl]piperidine-3-carboxylate
2-benzyl-8-(quinolin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetamide
2-(4-methoxyphenyl)-5-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}pyrimidine
4-{1-[3-(pyrrolidin-3-yl)benzoyl]piperidin-4-yl}pyridine
1-(3-methylpyridin-4-yl)-4-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1,4-diazepane
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl](1-methoxypropan-2-yl)amine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,1-dimethyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
(1R,5S,6S)-6-[(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]-3-azabicyclo[3.1.0]hexane
2-[1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]-6-methyl-1H-1,3-benzodiazole
1-(2-benzylmorpholin-4-yl)-2-phenoxyethan-1-one
2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-1-(morpholin-4-yl)ethan-1-one
3-chloro-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-6-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
8-benzyl-1-(2-methoxyethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-3-(propan-2-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]-1H-pyrazole-5-carboxamide
5-(3-fluorobenzoyl)-3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-ethylpiperazine
3-(1-methyl-1H-imidazol-2-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
4-{imidazo[1,2-a]pyrimidine-2-carbonyl}-1-methylpiperazin-2-one
8-(4-chloro-3-fluorobenzoyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-[({1-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}oxy)methyl]pyridine
N-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)-2-(2-methylphenyl)acetamide
1-[2-(4-fluorophenyl)piperidin-1-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
2-(3-methoxypropyl)-8-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{1-[(4-{[(3,4-dimethoxyphenyl)methyl](methyl)amino}quinazolin-2-yl)methyl]piperidin-4-yl}propan-1-ol
1-(1-ethylpiperidin-4-yl)-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
2-[5-(2,1,3-benzoxadiazol-5-yl)-4-phenyl-1H-imidazol-1-yl]-1-(pyridin-3-yl)ethan-1-ol
3-(1-methyl-1H-imidazol-2-yl)-1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidine
3-(2-methylphenoxy)-1-(5-methylthiophene-2-carbonyl)azetidine
5-(2-{2-[(5-chloropyridin-2-yl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
2-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(1-methyl-1H-1,3-benzodiazol-2-yl)-N-[2-(methylsulfanyl)phenyl]pyrrolidine-1-carboxamide
3-phenyl-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
N-benzyl-2-{2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}acetamide
2-[5-(5-chloro-7-methoxy-1-benzofuran-2-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-(2-{3-methyl-7-oxo-7H-[1,3]thiazolo[3,2-b][1,2,4]triazin-6-yl}phenyl)-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
N-(3-methoxypropyl)-1-(4-methylphenyl)-N-(1-methylpiperidin-4-yl)cyclopropane-1-carboxamide
methyl 4-(2-hydroxy-7-methylquinolin-3-yl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylate
2-methyl-8-{2-[methyl(phenyl)amino]acetyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(1S,9S)-11-[4-(pyridin-3-yl)pyrimidin-2-yl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
(3R,4R)-4-(azepan-1-yl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-ol
6-ethoxy-3-({methyl[(5-methyl-1,2-oxazol-3-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
5-[2-(adamantan-1-yl)acetyl]-N-methyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-4-methyl-1H-imidazole-5-carboxamide
1-methyl-3-(thiomorpholine-4-carbonyl)-N-[(3,4,5-trifluorophenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
8-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one