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2-{2-[1-(3-methylbenzenesulfonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
2-ethyl-4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-1-(propan-2-yl)piperazine
1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-(2-methoxyethoxy)piperidine
1-(4-{[(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}thiophen-2-yl)ethan-1-one
4-({5-[5-(4-methylphenyl)-1H-pyrazol-3-yl]-1,2,4-oxadiazol-3-yl}methyl)morpholine
benzyl[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amine
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N,5-dimethyl-N-(quinolin-5-ylmethyl)-1H-pyrazole-4-carboxamide
5-(2,6-dimethoxyphenyl)-3-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}-1,2,4-triazine
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
(1R,5R)-3-(2-fluorobenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
1-(cyclohexylmethyl)-N-methyl-5-[(1,2-oxazol-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-4-(4-methylphenoxy)piperidine-4-carboxamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{[4-(methylsulfanyl)phenyl]methyl}acetamide
(1R,5S,8R)-8-(dimethylamino)-N-[3-methyl-1-(2-methylphenyl)-1H-pyrazol-5-yl]-3-azabicyclo[3.2.1]octane-3-carboxamide
2-methyl-4-(4-{1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-imidazol-2-yl}phenyl)but-3-yn-2-ol
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-[3-(pyrazin-2-yl)propanoyl]-1,4-diazepan-2-one
3-acetamido-N-(4-methoxyphenyl)-5-({[(2-methylphenyl)methyl]amino}methyl)benzamide
4-[5-(methoxymethyl)thiophene-2-amido]-N-phenylpiperidine-1-carboxamide
1-ethyl-4-{[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-3-phenoxypropan-1-one
9-(2,5-dimethylbenzoyl)-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(2-methoxyethyl)-5-methyl-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-({4-[4-(dimethylamino)azepane-1-carbonyl]phenyl}(methyl)amino)ethan-1-ol
ethyl 1-[2-(4-methoxyphenyl)ethyl]-5-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-hydroxy-N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(thiophen-2-yl)pyrimidine-5-carboxamide
2-amino-4-(oxolan-3-yl)-6-[3-(propan-2-yloxy)phenyl]pyridine-3-carbonitrile
2-[1-(4-methylphenyl)cyclopropanecarbonyl]-2,7-diazaspiro[4.5]decan-6-one
3-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(trifluoromethyl)phenyl]urea
2-(3-methoxyphenoxy)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
(3aR,6aS)-1-oxo-5-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]acetyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(4-fluoro-2-methylphenyl)-2-{[1-(1H-imidazol-1-yl)propan-2-yl]amino}acetamide
4-[4-(1-carbamoylpiperidine-3-carbonyl)piperazin-1-yl]benzoic acid
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-(2H-1,3-benzodioxol-5-yl)-1-(furan-3-ylmethyl)piperidin-3-amine
N-tert-butyl-3-[2-(2H-indazol-2-yl)acetamido]-2-methylbenzamide
N,N-dimethyl-5-{[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(cyclopropylmethyl)-5-(piperidin-4-yl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
5-(hydroxymethyl)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}furan-2-carboxamide
2-[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]-1-phenylethan-1-ol
3-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
(1R,7S)-3-[(3-methoxyphenyl)methyl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[2-(2-chlorophenoxy)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
2-(1,2-benzoxazol-3-yl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}acetamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-(5-methyl-1,2-oxazol-3-yl)piperidine
2-methyl-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-(piperidin-4-yl)pyrimidin-4-amine
3-{[1-(4-methanesulfonylphenyl)propyl]carbamoyl}-5-methoxybenzoic acid
2-(1-ethylpiperidin-4-yl)-N-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}acetamide
3,5,7-trimethyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-indole-2-carboxamide
2-{1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1H-imidazol-2-yl}-4,5,6,7-tetrahydro-1,3-benzothiazole