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(2R,3R,6R)-5-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)pyridin-2-amine
10-methoxy-5-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-cyclopropyl-1-[(1s,4s)-4-{[(3,5-dimethoxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-[2-(4-cyclopentylphenyl)pyridine-4-carbonyl]morpholine
(4aS,8aR)-6-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
N-[1-(4-methanesulfonylphenyl)ethyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
1-methyl-1'-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
methyl 4-[({1-[4-(cyclopentylcarbamoyl)phenyl]piperidin-4-yl}amino)methyl]benzoate
2-(3-chloro-4-hydroxyphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}-N-(3-methoxyphenyl)piperidine-1-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidin-3-ol
9-(cyclopropylmethyl)-1-methyl-4-(morpholine-4-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
7-methyl-2-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-4H-chromen-4-one
2-(2-{[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]methyl}phenoxy)-N,N-dimethylacetamide
6-[3-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyrazine-2-carboxamide
1-[3-(dimethylamino)phenyl]-3-[1-(1-methyl-1H-imidazol-2-yl)butyl]urea
methyl 3-[(3S,4R)-4-(dimethylamino)-1-[(2-methoxyphenyl)methyl]piperidin-3-yl]propanoate
methyl (2R,4S)-1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-4-hydroxypiperidine-2-carboxylate
[(4aS,8aR)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-pentyl-decahydro-1,6-naphthyridin-4a-yl]methanol
2-[4-(2-amino-6-methylpyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-ethyl-1H-1,2,3-triazol-4-yl)acetamide
1-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
(3aR,7aS)-5-methyl-2-[3-(piperidine-1-carbonyl)pyridin-2-yl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
(2E)-1-{4-[2-(3-methoxyphenyl)-1-[methyl(pyridin-4-ylmethyl)amino]ethyl]piperidin-1-yl}-4-methylpent-2-en-1-one
2-[(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]acetic acid
3-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6-methylpyridazine
7-chloro-3-{[(2-methylpropyl)amino]methyl}-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
5-amino-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-phenyl-1H-pyrazole-3-carboxamide
1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1,4-diazepane-6-carboxylic acid
(1S,5R)-6-(2-fluoro-4-methylbenzoyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-(2-cyclohexylethyl)-N-methyl-N-(oxan-4-yl)-1H-1,2,3-triazole-4-carboxamide
N-(diphenylmethyl)-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl](methyl)[(5-methylfuran-2-yl)methyl]amine
N,N-diethyl-1-[(1s,4s)-4-[2-(3,4-dimethoxyphenyl)acetamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(2S,4R)-4-(3-chlorobenzamido)-N-[3-(1H-imidazol-1-yl)propyl]pyrrolidine-2-carboxamide
3-{[1-(2,2-difluorobutanoyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3aS,7aR)-5-methyl-2-[2-(3-methylphenoxy)acetyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
6-[(1S,5R)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carbonitrile
(2S,4S)-4-amino-N-ethyl-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidine-2-carboxamide
(3S,4S)-1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
N-tert-butyl-7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-cyclopentanecarbonyl-4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
N-(pyridin-3-ylmethyl)-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
(4aR,7aS)-1-methanesulfonyl-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
N-[(3-methylphenyl)methyl]-2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
(3S,4R)-N-(2,3-dichlorophenyl)-3-(dimethylamino)-4-propylpyrrolidine-1-carboxamide
(1S,3R)-3-amino-N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)cyclopentane-1-carboxamide
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-N,5-dimethyl-1,3,4-oxadiazole-2-carboxamide
methyl 4-{[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]carbamoyl}butanoate