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2-methyl-N-{2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]phenyl}furan-3-carboxamide
{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
4-(1-{1-[6-(propan-2-yl)pyrimidin-4-yl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[(5-methylfuran-2-yl)methyl]piperidine
1-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(methylsulfanyl)ethan-1-one
3-methyl-6-{5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1,2,4-oxadiazol-3-yl}pyridazine
2-({4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
5-[benzyl(methyl)amino]-2-[(3,4,5-trifluorophenyl)methyl]-2,3-dihydropyridazin-3-one
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[1-(1,3-thiazol-2-yl)ethyl]propanamide
1-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
(1H-1,3-benzodiazol-2-ylmethyl)[3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}benzamide
3-chloro-N-[2-(2-methoxy-5-{[4-(2-methylphenyl)piperazin-1-yl]methyl}phenoxy)ethyl]-2-methylbenzene-1-sulfonamide
2-[4-(1H-pyrazol-5-yl)phenyl]pyridin-3-ol
3-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-1,2-dimethyl-1H-indol-5-ol
3-hydroxy-1-(2-methoxyethyl)-3-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}piperidin-2-one
3-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-[2-(2-methoxyethoxy)phenyl]urea
2-({[(4,6-dimethylpyridin-3-yl)methyl]amino}methyl)-6-fluoroquinolin-4-ol
5-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-(1-{[(naphthalen-1-ylmethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)thiophene-3-carboxamide
3-{[7-(2,5-dimethylfuran-3-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine
N7-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-[1,2,4]triazolo[4,3-c]pyrimidine-5,7-diamine
1-(3-methoxyphenyl)-4-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperazin-2-one
(5S,9aS,9bS)-5-[5-(4-chlorophenyl)furan-2-yl]-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[7-(thiophene-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidin-4-ol
2-{1-[(2-cyclohexylpyrimidin-5-yl)methyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
N-(pyridin-4-ylmethyl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-pyrazol-1-yl)propan-1-one
methyl 5-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-{4-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}propanamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
2-(4-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
(1-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-4-(oxan-2-ylmethyl)piperidin-4-yl)methanol
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-methoxyquinoline-4-carboxamide
9-[(2S,3S)-2-amino-3-methylpentanoyl]-2-benzyl-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-3-azaspiro[5.5]undecan-9-amine
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(methylsulfanyl)acetamide
1-(2-methylpropyl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-5-oxopyrrolidine-3-carboxamide
3-[4-(adamantan-1-yl)piperazine-1-carbonyl]-2-(cyclopentylmethyl)-1,6-dimethyl-1,4-dihydropyridin-4-one
3-{2-[4-(hydroxymethyl)piperidin-1-yl]ethyl}-1-[3-(4-methylphenyl)phenyl]urea
5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,3-benzothiazol-2-amine
N-{1-[({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}benzamide
3-{5-[(2-phenylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
7-(cyclopropylmethyl)-2-(3-hydroxyazetidine-1-carbonyl)-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
3-(5-{1-[(2-fluoro-3-methoxyphenyl)methyl]pyrrolidin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-(3-phenylpropyl)propanamide
N-(cyclopropylmethyl)-N-propyl-1-benzofuran-3-carboxamide
(4aS,7aR)-1-(2-methylpropyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-[(2-methoxyphenyl)methyl]propanamide