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3-[2-(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)ethyl]-2,3-dihydro-1,3-benzoxazol-2-one
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
1-(cyclohexylmethyl)-N-methyl-5-[(2,2,2-trifluoroethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-benzyl-3-[2-(3-hydroxypiperidin-1-yl)-2-oxoethyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
2-{[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]amino}-N-[2-methyl-6-(propan-2-yl)phenyl]acetamide
4-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-5-methyl-2-phenyl-1,3-oxazole
3-(3-{7-[ethoxy(phenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-3-oxopropyl)-3,4-dihydroquinazolin-4-one
2-{2-[2-(3,5-dimethyl-1-benzofuran-2-yl)-1H-imidazol-1-yl]propyl}pyrazine
3-(4-methyl-1H-pyrazol-1-yl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
4-[(4-methylphenyl)methyl]-3-(2-oxo-2-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidin-1-yl}ethyl)piperazin-2-one
{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
5-methoxy-2-{4-[(4-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,4-dihydropyridin-4-one
4-chloro-N-{3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
4-[3-(2-methoxyethyl)-5-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
(4aR,7aS)-1-(3-methylbutanoyl)-4-(1,2-oxazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({3-methyl-7-[2-(7-methyl-2-oxo-2H-chromen-4-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
4-chloro-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
methyl 4-(3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}propanamido)butanoate
5-[1-(carbamoylmethyl)piperidine-4-carbonyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
5,6,7-trimethoxy-3-{[methyl(1-methylpyrrolidin-3-yl)amino]methyl}-1,2-dihydroquinolin-2-one
(2R,6R)-4-[(1-ethyl-1H-pyrazol-3-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-(1-methyl-1H-indazol-3-yl)-2-[5-(1-phenylcyclopropyl)-2H-1,2,3,4-tetrazol-2-yl]acetamide
N-(4-butanamido-3-methoxyphenyl)-4-oxo-1,4-dihydroquinoline-2-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(1H-indol-4-ylmethyl)piperidine-3-carboxamide
(4aS,7aR)-1-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-3-(1H-pyrazol-1-yl)propanamide
N4-[(1R)-1-(3-methoxyphenyl)ethyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
N-{[2-(dimethylamino)-7-(methylsulfanyl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-methylpropanamide
2-cyclopropyl-4-hydroxy-N-[(8-methoxyquinolin-5-yl)methyl]-N-methylpyrimidine-5-carboxamide
7-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carbonyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-3-fluoroimidazo[1,2-a]pyridine-2-carboxamide
6-{3-[1-(dimethylamino)ethyl]phenyl}-3,4-dihydroquinazolin-4-one
N-(2-methoxyethyl)-3-(2-methoxyphenyl)-N-{[6-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}propanamide
2-(ethoxymethyl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
1-[1-(2-methoxyethyl)piperidine-4-carbonyl]-4-phenylpiperidin-4-ol
[2-ethoxy-5-(1-methyl-1H-1,3-benzodiazol-2-yl)phenyl]methanol
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-4-(pyridin-4-yl)pyrimidin-2-amine
1-(2-methoxyphenyl)-4-{2-[4-(propan-2-yl)phenyl]acetyl}piperazin-2-one
4-(2,6-difluoro-4-methoxybenzoyl)-5-methyl-1-(3-methylphenyl)piperazin-2-one
{3-[2-(3-ethenylphenyl)-1H-imidazol-1-yl]phenyl}methanamine
2-(2-{[2-methoxy-1-(pyridin-2-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-[1-(2-phenylpropyl)piperidin-4-yl]-4-(pyrrolidine-1-carbonyl)piperidine
8-[(2-fluorophenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(benzyloxy)-1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
1-methyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-6-oxo-1,6-dihydropyridazine-3-carboxamide
4-{1-[2-(1H-imidazol-5-yl)ethyl]-3-phenyl-1H-1,2,4-triazol-5-yl}-1λ6-thiane-1,1-dione
N-{1-[1-(5-methoxyfuran-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-2-(trifluoromethyl)benzene-1-sulfonamide