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7-(1,3-benzothiazol-2-yl)-4-(2,4-dimethoxybenzoyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3R,5S)-N-[(1-ethylpyrrolidin-2-yl)methyl]-5-(morpholin-4-ylmethyl)-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
methyl(2-phenylethyl){[3-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1,2-oxazol-5-yl]methyl}amine
1-({5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]furan-2-yl}methyl)-4-methylpiperazine
5-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(2R,3R,6R)-5-(morpholine-4-sulfonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
2-ethoxy-6-[(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenol
5-ethoxy-N-(2-oxoazepan-3-yl)furan-2-carboxamide
1-(2-methoxyphenyl)-4-[1-(1,2,3-thiadiazole-4-carbonyl)piperidin-3-yl]piperazine
4-(pyrrolidine-1-carbonyl)-1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidine
5-cyclobutyl-N-[2-(3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]-1,3,4-oxadiazol-2-amine
8-(3-methyl-1H-pyrazole-5-carbonyl)-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1-phenyl-1H-1,2,3-triazole-5-carboxamide
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
5-(2-fluorobenzoyl)-2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-[7-(3-methyl-1H-pyrazole-5-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
4-(4-fluorophenyl)-1-(trimethylpyrimidin-4-yl)piperidin-4-ol
N-(3,5-dimethylphenyl)-6-[2-(2-methoxyphenoxy)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[2-(pyridin-3-yl)acetyl]piperidin-3-yl}propanamide
7-[cyclohexyl(methoxy)methyl]-4-(1,2,5-thiadiazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl)-3-methanesulfonylpropan-1-one
2-(1H-pyrazol-3-yl)-4-(3,3,3-trifluoropropyl)pyrimidine
N-[(3-chlorophenyl)methyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
(3R,4R)-4-ethyl-1-[2-(pyrrolidin-1-yl)-6-(trifluoromethyl)pyrimidin-4-yl]piperidine-3,4-diol
2-(3-{[({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)amino]methyl}phenoxy)ethan-1-ol
2-{4-[4-(benzyloxy)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}-N,N-diethylacetamide
3-(3-methoxyphenyl)-5-(thiophene-3-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
3-{[(4-hydroxy-6-methylquinolin-2-yl)methyl](methyl)amino}-1λ6-thiolane-1,1-dione
5-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}methyl)-N-ethylpyrimidin-2-amine
2-(6-methylpyridazin-3-yl)-N,N-bis(propan-2-yl)benzamide
3-({2-amino-3-ethyl-3H-imidazo[4,5-b]pyridin-6-yl}formamido)-N-cyclohexylpropanamide
N-methyl-5-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1-{3-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
4-{[3-(2-hydroxyethoxy)phenyl]methyl}-1-(2-methylphenyl)piperazin-2-one
N-(1-{1-[(3-ethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
2-methyl-5-(trifluoromethyl)-1-{1-[(2,3,4-trimethoxyphenyl)methyl]piperidin-4-yl}-1H-1,3-benzodiazole
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-3-(pyridin-4-yl)propanamide
2-amino-N-[2-(1,3-thiazol-4-yl)ethyl]-1,3-benzothiazole-5-carboxamide
2-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)-6-fluoroquinolin-4-ol
1-ethyl-6-methyl-3-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N,N-dimethyl-1-{1-[3-(2-methylphenyl)phenyl]piperidin-4-yl}piperidin-4-amine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
5-fluoro-N-[2-(1-methylpyrrolidin-2-yl)ethyl]quinazolin-4-amine
5-(piperidin-1-yl)-2-(pyridin-2-ylmethyl)-2,3-dihydropyridazin-3-one
N-methyl-N-[2-(morpholin-4-yl)propyl]cycloheptanamine
2-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[(2S)-1-methoxy-3-phenylpropan-2-yl]-2-(methylamino)pyrimidine-5-carboxamide
3-(2-methoxyethyl)-1-(2-phenylethyl)-8-(quinolin-8-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(cyclohexylmethyl)-3-[2-(methylsulfanyl)ethyl]-5-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepin-9-yl}-1H-1,2,4-triazole
4-methyl-3-[(2S)-2-(morpholine-4-carbonyl)pyrrolidine-1-carbonyl]benzene-1-sulfonamide